SCHEMBL11942285

SCHEMBL11942285

Cc1nc(C(N)=O)cc(N)c1F

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
GRM2 Q14416 10/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
NQO2 P16083 4/20 0.37
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CDK8 P49336 1/20 0.33
CDK19 Q9BWU1 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15449695 0.85 SMN1; SMN2 (0.39) LMNAPOLBKDM4EALDH1A1HPGD
SCHEMBL15440474 0.81 LMNA (0.45) LMNAGRM2NQO2SCN9A
SCHEMBL15452631 0.79 LMNA (0.44) LMNAGRM2NQO2ALDH1A1SCN9A
SCHEMBL11942291 0.71 LMNA (0.47) LMNAGRM2DPP4DPP8NQO2
SCHEMBL13824470 0.71 PIM1 (0.42) LMNAGRM2DPP4DPP8KDM4E
SCHEMBL29502454 0.69 TGFBR1 (0.42) LMNAGRM2DPP4DPP8KDM4E
SCHEMBL2827339 0.69 TGFBR1 (0.42) LMNAGRM2DPP4DPP8KDM4E
SCHEMBL23539404 0.69 LMNA (0.45) LMNAGRM2POLBKDM4EALDH1A1
SCHEMBL7718641 0.69 LMNA (0.54) LMNAGRM2NQO2POLB
SCHEMBL19462416 0.68 TERT (0.34) LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993772-B2 Process for the preparation of 4-amino-5-fluoro-3-halo-6-(substituted)picolinates DOW AGROSCIENCES, LLC. (US) 2015-03-31 US disclosed
US-8871943-B2 Process for the preparation of 4-amino-5-fluoro-3-halo-6-(substituted)picolinates DOW AGROSCIENCES, LLC. (US) 2014-10-28 US disclosed
US-20140206881-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES DOW AGROSCIENCES LLC (US) 2014-07-24 US disclosed
US-8754231-B2 Process for the preparation of 4-amino-5-fluoro-3-halo-6-(substituted)picolinates DOW AGROSCIENCES, LLC. (US) 2014-06-17 US disclosed
US-20140031556-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES DOW AGROSCIENCES LLC (US) 2014-01-30 US disclosed
US-20120190859-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES DOW AGROSCIENCES LLC (US) 2012-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140031556-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES CLIC4, NPEPPS, CYP4F3 LMNA 1962/4885GRM2 2379/4885DPP4 440/4885
US-20120190859-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES CYP4F3, CYP4F12, AFF4 LMNA 2800/4885GRM2 2134/4885DPP4 57/4885
US-20140206881-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-5-FLUORO-3-HALO-6-(SUBSTITUTED)PICOLINATES CYP4F3, CYP4F12, AFF4 LMNA 2800/4885GRM2 2134/4885DPP4 57/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.