SCHEMBL12010809

SCHEMBL12010809

CC(=O)N(C)Cc1ccc2c(c1)CN(C)CC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDK2 Q15119 1/20 0.41
MAOA P21397 4/20 0.40
MAOB P27338 4/20 0.40
QRFPR Q96P65 6/20 0.40
KCNH2 Q12809 2/20 0.40
CYP2D6 P10635 1/20 0.40
KCNE1 P15382 1/20 0.40
SCN5A Q14524 1/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
SLC6A4 P31645 1/20 0.39
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12010845 0.83 DRD2 (0.47) ALDH1A1POLBMAPTSMN1; SMN2PDK2
SCHEMBL12010846 0.83 ALDH1A1 (0.39) ALDH1A1POLBMAPTSMN1; SMN2PDK2
SCHEMBL19033381 0.81 RXRA (0.48) ALDH1A1POLBMAPTSMN1; SMN2PDK2
SCHEMBL1787581 0.78 HRH3 (0.48) CYP2D6
SCHEMBL1787583 0.78 MAPT (0.40) ALDH1A1POLBMAPTSMN1; SMN2PDK2
SCHEMBL12010814 0.78 OPRD1 (0.43) POLBMAPTQRFPRKCNH2CYP2D6
SCHEMBL14615342 0.77 ALDH1A1 (0.52) ALDH1A1MAOAMAOBDRD2DRD3
SCHEMBL5151266 0.77 SLC22A12 (0.49) ALDH1A1POLBMAPTMAOAMAOB
SCHEMBL12683145 0.76 MAOA (0.50) MAOAMAOBDRD2DRD3SLC6A4
SCHEMBL12010808 0.75 DRD2 (0.37) QRFPRKCNH2CYP2D6KCNE1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8252785-B2 Aryl sulfonamides as bradykinin-B1-receptor antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-28 US disclosed
US-8252785-B2 Aryl sulfonamides as bradykinin-B1-receptor antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-28 US disclosed