SCHEMBL12073915

SCHEMBL12073915

CC(=O)n1cc(CN2CCCCC2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
NCOR2 Q9Y618 1/20 0.51
HTR6 P50406 1/20 0.47
POLB P06746 2/20 0.47
RAD52 P43351 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PLK1 P53350 1/20 0.45
LMNA P02545 2/20 0.45
GLA P06280 1/20 0.45
ACHE P22303 1/20 0.45
HTR7 P34969 1/20 0.44
CREBBP Q92793 2/20 0.44
BRPF1 P55201 1/20 0.44
BRD9 Q9H8M2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084333 0.84 HTR7 (0.51) POLBMEN1KMT2ALMNAHTR7
SCHEMBL15081962 0.81 OPRL1 (0.48) HDAC8HDAC6POLBMEN1KMT2A
SCHEMBL807570 0.80 ALDH1A1 (0.47) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL12301581 0.79 CREBBP (0.52) POLBMEN1KMT2AGLACREBBP
SCHEMBL5961922 0.78 LMNA (0.69) HDAC8HDAC6HTR6LMNAGLA
SCHEMBL24331530 0.76 CREBBP (0.50) POLBMEN1KMT2AGLACREBBP
SCHEMBL23536600 0.75 HTR6 (0.51) HTR6POLBMEN1KMT2ACREBBP
SCHEMBL31432746 0.75 CDC25A (0.55) POLBPLK1LMNACREBBPBRPF1
SCHEMBL10359905 0.75 HTT (0.51) HDAC6HDAC10POLBMEN1KMT2A
SCHEMBL7182399 0.74 CREBBP (0.48) POLBMEN1KMT2AGLACREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163330-A1 NOVEL HETEROCYCLIC COMPOUNDS AS ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-12-29 WO disclosed