SCHEMBL807570

SCHEMBL807570

CCC[C@@H]1CCCN(Cc2cn(C(C)=O)c3ccccc23)C1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
BCHE P06276 3/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
ACHE P22303 2/20 0.40
HTR6 P50406 1/20 0.40
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084333 0.84 HTR7 (0.51) ALDH1A1MEN1KMT2APOLBTSHR
SCHEMBL15081962 0.82 OPRL1 (0.48) ALDH1A1MEN1KMT2AHDAC8HDAC6
SCHEMBL12073915 0.80 HDAC8 (0.51) MEN1KMT2AHDAC8HDAC6POLB
SCHEMBL807391 0.72 CHRNA7 (0.60) HDAC8HDAC6SMN1; SMN2TSHR
SCHEMBL12301581 0.72 CREBBP (0.52) ALDH1A1MEN1KMT2APOLBSMN1; SMN2
SCHEMBL12513821 0.71 CYP2D6 (0.59) ALDH1A1BCHEMEN1KMT2APOLB
SCHEMBL10212322 0.71 CYP2D6 (0.59) ALDH1A1BCHEMEN1KMT2APOLB
SCHEMBL807390 0.68 FAAH (0.44)
SCHEMBL12479944 0.67 CFD (0.60) ALDH1A1KMT2APOLBSMN1; SMN2
SCHEMBL13837069 0.67 CFD (0.60) ALDH1A1KMT2APOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed