SCHEMBL12142103

SCHEMBL12142103

CCc1ccc(-c2ccc(C(=O)O)cc2)c(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.63
AKR1C2 P52895 4/20 0.63
ALDH1A1 P00352 1/20 0.53
RXRA P19793 4/20 0.53
RXRB P28702 4/20 0.53
BCL2 P10415 1/20 0.52
SRD5A2 P31213 1/20 0.51
ADH5 P11766 1/20 0.48
FOLH1 Q04609 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RARB P10826 3/20 0.46
CYP2C8 P10632 1/20 0.46
RXRG P48443 3/20 0.45
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
S1PR1 P21453 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14791856 0.87 AKR1C3 (0.49) AKR1C3AKR1C2SRD5A2S1PR1
SCHEMBL12141744 0.86 NOTUM (0.49) AKR1C3AKR1C2SRD5A2S1PR1
SCHEMBL12142108 0.85 PLK1 (0.56) AKR1C3AKR1C2SRD5A2S1PR1
SCHEMBL12141580 0.83 KIF11 (0.53) AKR1C3AKR1C2RXRARXRBRXRG
SCHEMBL23302210 0.83 ADH5 (0.63) AKR1C3AKR1C2RXRARXRBSRD5A2
Hydrochloric Acid SCHEMBL28670680 0.82 ADH5 (0.61) AKR1C3AKR1C2RXRARXRBSRD5A2
SCHEMBL7368161 0.82 RORC (0.48) AKR1C3AKR1C2ALDH1A1NPC1RAB9A
SCHEMBL16255738 0.81 AKR1C3 (0.60) AKR1C3AKR1C2ALDH1A1RXRARXRB
SCHEMBL31236747 0.80 RXRA (0.58) AKR1C3AKR1C2RXRARXRBSRD5A2
SCHEMBL12141581 0.79 CHKA (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8394818-B2 Soluble mTOR complexes and modulators thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-12 US disclosed
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF MTOR, RICTOR, RPTOR AKR1C3 2849/4885AKR1C2 3156/4885ALDH1A1 4698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.