SCHEMBL12201435

SCHEMBL12201435

Cc1cccc(NS(=O)(=O)c2ccc(Cl)cc2)c1C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.67
METAP2 P50579 3/20 0.56
KEAP1 Q14145 1/20 0.55
NFE2L2 Q16236 1/20 0.55
CCR2 P41597 3/20 0.53
CCR1 P32246 1/20 0.53
LMNA P02545 2/20 0.51
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.51
HTT P42858 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
GPR27 Q9NS67 1/20 0.50
ACLY P53396 1/20 0.50
FLT1 P17948 1/20 0.50
FLT4 P35916 1/20 0.50
KDR P35968 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14267572 0.89 ALDH1A1 (0.67) ALDH1A1METAP2CCR2CCR1LMNA
SCHEMBL12200962 0.89 POLB (0.60) ALDH1A1METAP2KEAP1NFE2L2LMNA
SCHEMBL2478529 0.84 KEAP1 (0.68) ALDH1A1KEAP1NFE2L2LMNAGAA
SCHEMBL12200867 0.81 KCNA5 (0.61) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL7562043 0.81 ALDH1A1 (1.00) ALDH1A1KEAP1CCR2LMNAKDM4E
SCHEMBL12200806 0.79 LMNA (0.56) ALDH1A1KEAP1NFE2L2LMNAGAA
SCHEMBL12200963 0.79 ACLY (0.78) ALDH1A1METAP2CCR2CCR1LMNA
SCHEMBL12202024 0.79 KCNA5 (0.66) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL12202030 0.79 KCNA5 (0.64) ALDH1A1
SCHEMBL12200779 0.77 CCR2 (0.73) ALDH1A1METAP2CCR2CCR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385820-B1 ANTHRANILIC ACID AMIDES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS ANTIARRHYTHMIA AGENTS, AND PHARMACEUTICAL PREPARATIONS THEREOF SANOFI AVENTIS DEUTSCHLAND (DE) 2011-10-12 EP disclosed
US-7332608-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-02-19 US disclosed
US-7332608-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-02-19 US disclosed
US-7235690-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed
US-7235690-B2 Anthranilamides and methods of their use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-05-24 US disclosed
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117807-A1 ANTHRANILAMIDES AND METHODS OF THEIR USE KCNH1, KCNH2, KCNJ2 ALDH1A1 1053/4885METAP2 4099/4885KEAP1 1722/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.