Ganomycin B

Ganomycin B

SCHEMBL12249396

CC(C)=CCC/C(C)=C/CC/C(=C/Cc1cc(O)ccc1O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.65
PTGS2 P35354 2/20 0.56
ACHE P22303 1/20 0.54
CTSK P43235 1/20 0.48
ALOX5 P09917 1/20 0.48
ALOX15 P16050 1/20 0.48
MAOB P27338 2/20 0.46
HTT P42858 1/20 0.46
APP P05067 2/20 0.45
PTPN1 P18031 1/20 0.45
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768674 1.00 BACE1 (0.65) BACE1PTGS2ACHECTSKALOX5
Ganomycin B SCHEMBL30164283 1.00 BACE1 (0.65) BACE1PTGS2ACHECTSKALOX5
Ganomycin B SCHEMBL6764577 1.00 BACE1 (0.65) BACE1PTGS2ACHECTSKALOX5
Ganomycin B SCHEMBL7074168 1.00 BACE1 (0.65) BACE1PTGS2ACHECTSKALOX5
Ganomycin A SCHEMBL6765493 0.92 PTGS2 (0.67) BACE1PTGS2ACHECTSKALOX5
SCHEMBL6764548 0.92 PTGS2 (0.67) BACE1PTGS2ACHECTSKALOX5
Ganomycin A SCHEMBL7074132 0.92 PTGS2 (0.67) BACE1PTGS2ACHECTSKALOX5
SCHEMBL6761207 0.92 PTGS2 (0.67) BACE1PTGS2ACHECTSKALOX5
Ganomycin A SCHEMBL1839019 0.92 PTGS2 (0.67) BACE1PTGS2ACHECTSKALOX5
SCHEMBL6764592 0.91 BACE1 (0.54) BACE1PTGS2ACHECTSKALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10441562-B2 Aromatic farnesyl compound and application thereof INSTITUTE OF MICROBIOLOGY, CHINESE ACADEMY OF SCIENCES (CN) 2019-10-15 US disclosed
WO-2018014660-A1 USE OF AROMATIC FARNESYL COMPOUNDS 中国科学院微生物研究所 2018-01-25 WO disclosed
US-20170224651-A1 AROMATIC FARNESYL COMPOUND AND APPLICATION THEREOF INSTITUTE OF MICROBIOLOGY, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-10 US disclosed
US-20170224651-A1 AROMATIC FARNESYL COMPOUND AND APPLICATION THEREOF INSTITUTE OF MICROBIOLOGY, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-10 US disclosed
WO-2016173274-A1 AROMATIC FARNESYL COMPOUND AND APPLICATION THEREOF 中国科学院微生物研究所 2016-11-03 WO disclosed
US-8466311-B2 Neuroprotective compositions and methods SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2013-06-18 US disclosed
US-8466311-B2 Neuroprotective compositions and methods SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2013-06-18 US disclosed
US-20120296112-A1 Neuroprotective Compositions and Methods NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-11-22 US disclosed
US-20120296112-A1 Neuroprotective Compositions and Methods NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-11-22 US disclosed
US-8022246-B2 Neuroprotective compositions and methods THE BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2011-09-20 US disclosed
US-8022246-B2 Neuroprotective compositions and methods THE BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2011-09-20 US disclosed
US-20090042980-A1 Neuroprotective compositions and methods BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2009-02-12 US disclosed
US-20090042980-A1 Neuroprotective compositions and methods BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2009-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10441562-B2 Aromatic farnesyl compound and application thereof HMGCR, PYGL, TGFB1 BACE1 509/4885PTGS2 1779/4885ACHE 2541/4885
US-20090042980-A1 Neuroprotective compositions and methods KEAP1, NFE2L2, NQO1 BACE1 176/4885PTGS2 21/4885ACHE 1738/4885
US-20120296112-A1 Neuroprotective Compositions and Methods KEAP1, NFE2L2, NQO1 BACE1 176/4885PTGS2 21/4885ACHE 1738/4885
US-20170224651-A1 AROMATIC FARNESYL COMPOUND AND APPLICATION THEREOF HMGCR, PYGL, TGFB1 BACE1 509/4885PTGS2 1779/4885ACHE 2541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.