Dextrorphan

Dextrorphan

SCHEMBL122564

CN1CC[C@@]23CCCC[C@@H]2[C@@H]1Cc1ccc(O)cc13.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1

The experimentally established mechanism targets of Dextrorphan. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 6/20 0.98
OPRD1 P41143 5/20 1.00
GRIN1 Q05586 8/20 0.98
GRIN2A Q12879 8/20 0.98
GRIN2D O15399 7/20 0.98
GRIN3B O60391 7/20 0.98
GRIN2B Q13224 7/20 0.98
GRIN2C Q14957 7/20 0.98
GRIN3A Q8TCU5 7/20 0.98
OPRK1 P41145 5/20 0.98
SLC22A1 O15245 3/20 0.98
SLC6A4 P31645 3/20 0.98
MRGPRX2 Q96LB1 3/20 0.98
CYP2D6 P10635 3/20 0.98
SLC6A2 P23975 3/20 0.98
SCN1A P35498 2/20 0.98
SCN2A Q99250 2/20 0.98
SCN3A Q9NY46 2/20 0.98
ADRA2A P08913 2/20 0.98
KCNH2 Q12809 2/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levorphanol SCHEMBL442528 1.00 OPRD1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL32667565 1.00 OPRD1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL24335 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL3495833 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL16310821 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL12232844 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL21095576 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL22722062 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Dextrorphan SCHEMBL20535964 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B
Levorphanol SCHEMBL22791693 0.99 GRIN1 (1.00) OPRD1GRIN1GRIN2AGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 230 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-12605333-B2 Modified release drug powder composition comprising gastro-retentive raft forming systems having trigger pulse drug release TRIS PHARMA, INC. (US) 2026-04-21 US disclosed
US-20260098013-A1 Stereoisomer Conjugates of Dextrorphan ZEVRA THERAPEUTICS INC (US) 2026-04-09 US disclosed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
US-20250339367-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-06 US disclosed
US-12403090-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-09-02 US disclosed
WO-1999030690-A1 ORAL DELIVERY FORMULATION AXIA THERAPEUTICS, INC. (US) 1999-06-24 WO disclosed
WO-1999026620-A1 CHOLINE ESTERS OF FATTY ACIDS AND THEIR USE IN THE TREATMENT OF STROKE PROTARGA, INC. (US) 1999-06-03 WO disclosed
EP-0909183-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES Neuromedica, Inc. (US) 1999-04-21 EP disclosed
WO-1998050044-A1 COMPOSITION AND METHOD COMBINING AN ANTIDEPRESSANT WITH AN NMDA RECEPTOR ANTAGONIST, FOR TREATING NEUROPATHIC PAIN ALGOS PHARMACEUTICAL CORPORATION (US) 1998-11-12 WO disclosed
US-5795909-A ANTICARCINOGENIC AND ANTITUMOR AGENTS; BREAST, COLON, OVARIANCANCERS NEUROMEDICA, INC. (US) 1998-08-18 US disclosed
WO-1997044063-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES NEUROMEDICA, INC. (US) 1997-11-27 WO disclosed
US-5019579-A Antitussive Agents PRODOTTI FORMETI S.R.L. (IT) 1991-05-28 US disclosed
EP-0219896-A1 Pharmaceutical compositions on the basis of dextrorphan for intranasal application PRODOTTI FORMENTI S.r.l. (IT) 1987-04-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12605333-B2 Modified release drug powder composition comprising gastro-retentive raft forming systems having trigger pulse drug release SI, GRPR, FABP2 OPRM1 735/4885OPRD1 550/4885GRIN1 334/4885
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES SORD, SLC6A13, CACNA1A OPRM1 1993/4885OPRD1 2462/4885GRIN1 2190/4885
US-20260098013-A1 Stereoisomer Conjugates of Dextrorphan OPRM1, OPRD1, OPRK1 OPRM1 1/4885OPRD1 2/4885GRIN1 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.