SCHEMBL12366179

SCHEMBL12366179

[C-]#[N+]CC(=O)NCc1cccc(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.46
MAOB P27338 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
KDM4E B2RXH2 3/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 1/20 0.40
RIPK1 Q13546 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
MAPK1 P28482 1/20 0.38
PDE10A Q9Y233 1/20 0.38
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366133 0.88 HPGD (0.54) SMN1; SMN2HPGDALDH1A1MEN1KMT2A
SCHEMBL12366166 0.86 P2RX7 (0.49) P2RX7
SCHEMBL12366161 0.79 RIPK1 (0.38) P2RX7KDM4ERIPK1CHRM4
SCHEMBL3558621 0.77 P2RX7 (0.51) P2RX7MAOBSMN1; SMN2HPGDALDH1A1
SCHEMBL12366210 0.76 ERCC1 (0.40) P2RX7SMN1; SMN2HPGDALDH1A1MEN1
SCHEMBL12366173 0.76 P2RX7 (0.52) P2RX7SMN1; SMN2HPGDALDH1A1MEN1
SCHEMBL12366170 0.76 CNR1 (0.46) P2RX7SMN1; SMN2ALDH1A1LMNARAB9A
SCHEMBL12366196 0.76 KMT2A (0.58) P2RX7SMN1; SMN2HPGDMEN1KMT2A
SCHEMBL2264097 0.76 MCL1 (0.54) P2RX7MAOBSMN1; SMN2HPGDALDH1A1
SCHEMBL12366137 0.76 P2RX7 (0.50) P2RX7MAOBMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed