SCHEMBL12366181

SCHEMBL12366181

[C-]#[N+]CC(=O)NCc1ccccc1Br

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
MAPT P10636 1/20 0.50
RIPK1 Q13546 1/20 0.50
P2RX7 Q99572 4/20 0.48
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
ALDH1A1 P00352 2/20 0.45
LMNA P02545 1/20 0.44
ANPEP P15144 1/20 0.44
TP53 P04637 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
THRB P10828 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366133 0.81 HPGD (0.54) KMT2ANPC1RAB9AMAPTRIPK1
SCHEMBL12366141 0.81 NPC1 (0.62) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL12366090 0.81 ALDH1A1 (0.57) KMT2ANPC1RAB9AP2RX7ALDH1A1
SCHEMBL12366196 0.78 KMT2A (0.58) KMT2AMAPTP2RX7CA2LMNA
SCHEMBL2905338 0.78 RIPK1 (0.62) KMT2ANPC1RAB9AMAPTRIPK1
SCHEMBL30259906 0.78 RIPK1 (0.62) KMT2ANPC1RAB9AMAPTRIPK1
SCHEMBL12366112 0.77 EPHX2 (0.51) KMT2AP2RX7MEN1
SCHEMBL11591975 0.76 GAA (0.59) KMT2ARAB9AMAPTALDH1A1LMNA
SCHEMBL2456852 0.75 KMT2A (0.58) KMT2ANPC1RAB9AMAPTRIPK1
SCHEMBL12366179 0.75 P2RX7 (0.46) KMT2ANPC1RAB9ARIPK1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed