SCHEMBL12366395

SCHEMBL12366395

[C-]#[N+]c1c(C(F)(F)F)cc(-c2ccccc2)n(Cc2ccc(Cl)c(Cl)c2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 11/20 0.44
PKM P14618 1/20 0.41
PGR P06401 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
EPHX2 P34913 1/20 0.38
PPARG P37231 1/20 0.38
DCTPP1 Q9H773 1/20 0.37
CNR1 P21554 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
SRC P12931 1/20 0.36
PRKACA P17612 1/20 0.36
PRKACG P22612 1/20 0.36
PRKACB P22694 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366320 0.90 KDM4E (0.47) KDM4EHPGDEPHX2PPARGDCTPP1
SCHEMBL12366238 0.90 DCTPP1 (0.42) KDM4EHPGDPPARGDCTPP1CNR1
SCHEMBL12366212 0.90 CNR1 (0.44) KDM4EHPGDPPARGDCTPP1CNR1
SCHEMBL12366415 0.89 CCR2 (0.41) CCR2PKMEPHX2PPARGITGB1
SCHEMBL12366308 0.88 RXRA (0.43) KDM4EHPGDEPHX2DCTPP1CNR1
SCHEMBL12366275 0.88 CFTR (0.42) KDM4EHPGDPPARGDCTPP1CNR1
SCHEMBL12366313 0.87 CNR1 (0.38) KDM4EHPGDDCTPP1CNR1ITGB1
SCHEMBL12366245 0.87 CNR1 (0.43) KDM4EHPGDDCTPP1CNR1ITGB1
SCHEMBL12366485 0.86 HPGD (0.40) KDM4EHPGDPPARGDCTPP1CNR1
SCHEMBL12366421 0.86 RXRA (0.39) KDM4EHPGDPPARGDCTPP1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed