SCHEMBL1239155

SCHEMBL1239155

C=CC(=O)OC(C#N)Cc1ccc(C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.38
DPP4 P27487 4/20 0.38
FAP Q12884 2/20 0.38
DPP8 Q6V1X1 2/20 0.38
DPP9 Q86TI2 2/20 0.38
DPP7 Q9UHL4 2/20 0.38
MAOB P27338 1/20 0.38
SAE1 Q9UBE0 1/20 0.37
UBA2 Q9UBT2 1/20 0.37
HTT P42858 1/20 0.37
CTSC P53634 6/20 0.37
KCNH2 Q12809 3/20 0.37
CTBP2 P56545 1/20 0.36
LTB4R Q15722 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
RAB9A P51151 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
CYP2A6 P11509 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4906568 0.83 MAOB (0.45) ACACBMAOBSAE1UBA2HTT
SCHEMBL3451969 0.78 LDHA (0.51) HTT
SCHEMBL3452224 0.76 HCAR2 (0.41) CTSK
SCHEMBL587685 0.74 GAA (0.47) MAOBSAE1UBA2HTTCTBP2
SCHEMBL3451136 0.74 TAAR1 (0.46) HTTCTBP2RAB9AMMP13
SCHEMBL27582698 0.72 THRB (0.50) SAE1UBA2HTTKCNH2CTBP2
SCHEMBL6778872 0.72 GSK3B (0.44) ACACBDPP4FAPDPP8DPP9
SCHEMBL10073623 0.71 MMP3 (0.44) RAB9AMMP12MMP13
SCHEMBL529992 0.70 TSHR (0.38)
SCHEMBL343191 0.70 THRB (0.50) RAB9AMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3392235-B1 BISCHLOROFORMATE COMPOSITION, BISCHLOROFORMATE COMPOSITION PRODUCTION METHOD, BISCHLOROFORMATE COMPOSITION CONTAINING SOLUTION, POLYCARBONATE RESIN, POLYCARBONATE RESIN PRODUCTION METHOD, COATING LIQUID, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND ELECTROPHOTOGRAPHIC DEVICE IDEMITSU KOSAN CO (JP) 2020-04-29 EP disclosed
US-10241427-B2 Polycarbonate copolymer, coating solution, electrophotographic photoreceptor, and electric device IDEMITSU KOSAN CO., LTD. (JP) 2019-03-26 US disclosed
US-20180364598-A1 BISCHLOROFORMATE COMPOSITION, BISCHLOROFORMATE COMPOSITION PRODUCTION METHOD, BISCHLOROFORMATE COMPOSITION-CONTAINING SOLUTION, POLYCARBONATE RESIN, POLYCARBONATE RESIN PRODUCTION METHOD, COATING LIQUID, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND ELECTROPHOTOGRAPHIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2018-12-20 US disclosed
EP-3392235-A1 BISCHLOROFORMATE COMPOSITION, BISCHLOROFORMATE COMPOSITION PRODUCTION METHOD, BISCHLOROFORMATE COMPOSITION CONTAINING SOLUTION, POLYCARBONATE RESIN, POLYCARBONATE RESIN PRODUCTION METHOD, COATING LIQUID, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND ELECTROPHOTOGRAPHIC DEVICE Idemitsu Kosan Co., Ltd (JP) 2018-10-24 EP disclosed
EP-3006483-B1 POLYCARBONATE COPOLYMER, COATING LIQUID USING SAME, MOLDED BODY, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO (JP) 2018-01-03 EP disclosed
EP-2447299-B1 POLYCARBONATE COPOLYMER, COATING LIQUID USING SAME, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO (JP) 2017-11-29 EP disclosed
US-20170075237-A1 POLYCARBONATE COPOLYMER, COATING SOLUTION, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND ELECTRIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2017-03-16 US disclosed
US-9551946-B2 Polycarbonate copolymer, coating liquid using same, molded body, and electrophotographic photosensitive body IDEMITSU KOSAN CO., LTD. (JP) 2017-01-24 US disclosed
EP-2862887-B1 POLYCARBONATE COPOLYMER, COATING LIQUID USING SAME, AND ELECTROPHOTOGRAPHIC PHOTORECEPTOR IDEMITSU KOSAN CO (JP) 2016-12-14 EP disclosed
US-9458291-B2 Polycarbonate copolymer IDEMITSU KOSAN CO., LTD. (JP) 2016-10-04 US disclosed
US-8043775-B2 Electrophotographic photosensitive body IDEMITSU KOSAN CO., LTD. (JP) 2011-10-25 US disclosed
EP-2378363-A1 POLYCARBONATE RESIN, COATING LIQUID CONTAINING SAME, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY Idemitsu Kosan Co., Ltd. (JP) 2011-10-19 EP disclosed
US-7893185-B2 Polycarbonate copolymer, method for producing the same, molded body, optical material, and electrophotographic photosensitive body IDEMITSU KOSAN CO., LTD. (JP) 2011-02-22 US disclosed
US-20100324209-A1 POLYCARBONATE COPOLYMER, METHOD FOR PRODUCING THE SAME, MOLDED BODY, OPTICAL MATERIAL, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO., LTD. (JP) 2010-12-23 US disclosed
US-20100233603-A1 POLYCARBONATE POLYMER, COATING LIQUID, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO., LTD. (JP) 2010-09-16 US disclosed
US-20090326184-A1 POLYCARBONATE COPOLYMER, METHOD FOR PRODUCING THE SAME, MOLDED BODY, OPTICAL MATERIAL, AND ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO., LTD. (JP) 2009-12-31 US disclosed
US-20090081569-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE BODY IDEMITSU KOSAN CO., LTD. (JP) 2009-03-26 US disclosed
EP-0780363-B1 Bisazo-benzofuran compounds, their use as charge carrier generating compounds SHARP KK (JP) 2001-09-26 EP disclosed
US-5853930-A Electrophotographic photoconductors using bisazo compounds SHARP KABUSHIKI KAISHA (JP) 1998-12-29 US disclosed
EP-0780363-A1 Bisazo-benzofuran compounds, their use as charge carrier generating compounds and intermediates for their preparation SHARP KABUSHIKI KAISHA (JP) 1997-06-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180364598-A1 BISCHLOROFORMATE COMPOSITION, BISCHLOROFORMATE COMPOSITION PRODUCTION METHOD, BISCHLOROFORMATE COMPOSITION-CONTAINING SOLUTION, POLYCARBONATE RESIN, POLYCARBONATE RESIN PRODUCTION METHOD, COATING LIQUID, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, AND ELECTROPHOTOGRAPHIC DEVICE NR2E3, REV1, PBRM1 ACACB 3581/4885DPP4 4693/4885FAP 4535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.