SCHEMBL124147

SCHEMBL124147

CCOC(=O)C1=NOC(c2ccccc2)(c2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
KDM4E B2RXH2 2/20 0.47
RECQL P46063 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
GAA P10253 4/20 0.44
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 3/20 0.42
OPRM1 P35372 4/20 0.41
NPSR1 Q6W5P4 3/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 2/20 0.40
GLA P06280 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7640011 1.00 MAPT (0.47) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL6051256 0.94 LMNA (0.44) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL342177 0.93 MAPT (0.43) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL694567 0.89 LMNA (0.48) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL29205863 0.84 MAPT (0.46) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL28401713 0.83 LMNA (0.42) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL6051255 0.82 MAPT (0.38) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL17584752 0.82 ALDH1A1 (0.41) MAPTKDM4ERECQLTDP1KMT2A
SCHEMBL29216618 0.81 PDCD1 (0.41) MAPTKDM4EKMT2ATSHRHSD17B10
SCHEMBL2469272 0.80 OPRM1 (0.40) MAPTKDM4EKMT2AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8850 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3947350-B1 SUBSTITUTED 2-HETEROARYL AMINOBENZENES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS BAYER AG (DE) 2026-05-27 EP claimed
EP-4742896-A1 HERBICIDE COMPOSITIONS COMPRISING MALONAMIDES AND SAFENERS FOR SELECTIVE WEED CONTROL IN CROPS BASF SE (DE) 2026-05-20 EP claimed
US-12610950-B2 Method for weed control in lawn or turf DISCOVERY PURCHASER CORPORATION (US) 2026-04-28 US claimed
US-12599136-B2 Substituted isophthalic acid diamides and their use as herbicides BAYER AKTIENGESELLSCHAFT (DE) 2026-04-14 US claimed
US-12593846-B2 Combinations of triazolone herbicides with safeners UPL Corporation Limited (MU) 2026-04-07 US claimed
US-20260068885-A1 HERBICIDAL COMPOSITIONS BAYER AG (DE) 2026-03-12 US claimed
US-20260060254-A1 HERBICIDAL COMPOSITIONS BAYER AG (DE) 2026-03-05 US claimed
US-20260000082-A1 STABILIZED LIQUID HERBICIDE FORMULATION OF HIGH-LOAD PYRASULFOTOLE ADAMA AGAN LTD. (IL) 2026-01-01 US claimed
US-12509445-B2 Herbicidally active 4-cyclopropyl-6-[4-(trifluormethyl)pyrazol-1-yl)]pyrimidines BAYER AKTIENGESELLSCHAFT (DE) 2025-12-30 US claimed
US-12492173-B2 Herbicidal substituted N-tetrazolyl aryl carboxamides BAYER AKTIENGESELLSCHAFT (DE) 2025-12-09 US claimed
WO-2002001957-A1 ARYL SULFONYL AMINO CARBONYL TRIAZOLE BASED SELECTIVE HERBICIDES BAYER CROPSCIENCE AG (DE) 2002-01-10 WO claimed
WO-2001089301-A1 SELECTIVE HETEROARYLOXY-ACETAMIDE-BASED HERBICIDES BAYER CROPSCIENCE AG (DE) 2001-11-29 WO claimed
WO-2001039597-A2 N-ARYL-URACILE-BASED HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-06-07 WO claimed
WO-2001037652-A2 CARBAMOYL TRIAZOLINONE-BASED HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-05-31 WO claimed
WO-2001035741-A2 SYNERGISTIC HERBICIDAL ACTIVE SUBSTANCE COMBINATIONS BAYER AKTIENGESELLSCHAFT (DE) 2001-05-25 WO claimed
WO-2001035740-A2 SELECTIVE HERBICIDES BASED UPON 2,6-DISUBSTITUTED PYRIDINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2001-05-25 WO claimed
WO-2001024633-A2 SELECTIVE HERBICIDES BASED ON PYRIMIDINE-DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2001-04-12 WO claimed
WO-2001022819-A1 SELECTIVE HERBICIDES ON THE BASIS OF N-ARYL-TRIAZOLINE(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 2001-04-05 WO claimed
WO-2001017350-A1 NEW HERBICIDAL COMPOSITIONS AVENTIS CROPSCIENCE UK LIMITED (GB) 2001-03-15 WO claimed
US-6124240-A Combinations of sulfonylurea herbicides and safeners HOECHST AGREVO GMBH (DE) 2000-09-26 US claimed