SCHEMBL12438545

SCHEMBL12438545

CCOC(=O)[C@H](CSSC[C@H](NC(=O)OC(C)(C)C)C(=O)OCC)NC(=O)OC(C)(C)C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.72
CYP2C9 P11712 1/20 0.72
CYP2C19 P33261 1/20 0.72
HTT P42858 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.64
ALDH1A1 P00352 3/20 0.57
MAPT P10636 3/20 0.57
KDM4E B2RXH2 1/20 0.53
GAA P10253 1/20 0.53
PKM P14618 1/20 0.53
HPGD P15428 1/20 0.53
ALOX12 P18054 1/20 0.53
CTSK P43235 6/20 0.46
CTSS P25774 5/20 0.46
PPARG P37231 3/20 0.41
PPARA Q07869 3/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CTSL P07711 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16626925 0.93 CYP1A2 (0.64) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL13138386 0.90 CYP1A2 (0.72) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL15608320 0.88 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL18167329 0.88 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL28777391 0.88 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL12934327 0.88 CYP1A2 (0.77) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL29739948 0.87 SMN1; SMN2 (0.65) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL28943389 0.87 SMN1; SMN2 (0.65) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL25003377 0.87 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2
SCHEMBL9679571 0.87 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040261-B2 Compounds as L-cystine crystallization inhibitors and uses thereof NEW YORK UNIVERSITY (US) 2015-05-26 US disclosed
US-20150099806-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NEW YORK UNIVERSITY 2015-04-09 US disclosed
US-8916609-B2 Compounds as L-cystine crystallization inhibitors and uses thereof NEW YORK UNIVERSITY (US) 2014-12-23 US disclosed
US-8916609-B2 Compounds as L-cystine crystallization inhibitors and uses thereof NEW YORK UNIVERSITY (US) 2014-12-23 US disclosed
US-8450089-B2 Compounds as L-cystine crystallization inhibitors and uses thereof NEW YORK UNIVERSITY (US) 2013-05-28 US disclosed
US-8450089-B2 Compounds as L-cystine crystallization inhibitors and uses thereof NEW YORK UNIVERSITY (US) 2013-05-28 US disclosed
US-20120316236-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NEW YORK UNIVERSITY 2012-12-13 US disclosed
US-20120316236-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NEW YORK UNIVERSITY 2012-12-13 US disclosed
US-20110177173-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-07-21 US disclosed
US-20110177173-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-07-21 US disclosed
WO-2011062640-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF NEW YORK UNIVERSITY (US) 2011-05-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150099806-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF ATP6V1B1, GLS, REN CYP1A2 2776/4885CYP2C9 1461/4885CYP2C19 2452/4885
US-20110177173-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF GLS, PKD1, CLIC1 CYP1A2 2598/4885CYP2C9 1819/4885CYP2C19 2603/4885
US-20120316236-A1 COMPOUNDS AS L-CYSTINE CRYSTALLIZATION INHIBITORS AND USES THEREOF ATP6V1B1, GLS, REN CYP1A2 2776/4885CYP2C9 1461/4885CYP2C19 2452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.