Ripisartan

Ripisartan

SCHEMBL12465608

CCCc1nc(C)n2[nH]c(=O)nc2c1Cc1ccc(-c2ccccc2-c2nn[nH]n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ripisartan SCHEMBL489673 0.85 AGTR1 (0.73) AGTR1
SCHEMBL9308944 0.81 AGTR1 (0.69) AGTR1
SCHEMBL9308977 0.80 AGTR1 (0.66) AGTR1
SCHEMBL22800020 0.77 AGTR1 (0.63) AGTR1
SCHEMBL9309816 0.77 AGTR1 (0.63) AGTR1
SCHEMBL9310003 0.76 AGTR1 (0.62) AGTR1
SCHEMBL9308892 0.76 AGTR1 (0.62) AGTR1
SCHEMBL9308916 0.76 AGTR1 (0.61) AGTR1
SCHEMBL9309944 0.75 AGTR1 (0.60) AGTR1
SCHEMBL9309293 0.74 AGTR1 (0.59) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113056465-B Tetrahydropyrane (THP) -substituted bicyclic pyrimidinedione compounds 迈奥卡迪亚公司 2025-01-28 CN claimed
EP-3873904-B1 TETRAHYDROPYRAN (THP)-SUBSTITUTED BICYCLIC-PYRIMIDINEDIONE COMPOUNDS MYOKARDIA INC (US) 2024-07-10 EP claimed
US-20220340569-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES MYOKARDIA INC (US) 2022-10-27 US claimed
EP-4054588-A1 METHODS OF TREATMENT WITH MYOSIN MODULATOR MyoKardia, Inc. (US) 2022-09-14 EP claimed
US-20220106314-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES MYOKARDIA INC (US) 2022-04-07 US claimed
EP-4736855-A2 TETRAHYDROPYRAN (THP)-SUBSTITUTED BICYCLIC-PYRIMIDINEDIONE COMPOUNDS MyoKardia, Inc. (US) 2026-05-06 EP disclosed
US-12616697-B2 Methods of treatment with myosin modulator MyoKardia, Inc. (US) 2026-05-05 US disclosed
EP-4464321-B1 TETRAHYDROPYRAN (THP)-SUBSTITUTED BICYCLIC-PYRIMIDINEDIONE COMPOUNDS MYOKARDIA INC (US) 2026-01-21 EP disclosed
US-20250339395-A1 COMPOUNDS CONTAINING S-N-VALERYL-N-{[2'-(1H-TETRAZOLE-5-YL)-BIPHENYL-4-YL]-METHYL}-VALINE AND (2R,4S)-5-BIPHENYL-4-YL-4-(3-CARBOXY-PROPIONYLAMINO)-2-METHYL-PENTANOIC ACID ETHYL ESTER MOIETIES AND CATIONS NOVARTIS PHARMACEUTICALS CORP (US) 2025-11-06 US disclosed
US-20250325531-A1 TREATMENT OF SYSTOLIC DYSFUNCTION MyoKardia, Inc. (US) 2025-10-23 US disclosed
US-20250282779-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES MYOKARDIA INC (US) 2025-09-11 US disclosed
US-20250241903-A1 TREATMENT OF SYSTOLIC DYSFUNCTION MYOKARDIA INC (US) 2025-07-31 US disclosed
WO-2022047004-A1 METHODS OF TREATMENT WITH MYOSIN MODULATOR MyoKardia, Inc. (US) 2022-03-03 WO disclosed
US-8569528-B2 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides NOVARTIS AG (CH) 2013-10-29 US disclosed
US-20120330026-A1 PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES NOVARTIS AG (CH) 2012-12-27 US disclosed
US-20110184187-A1 PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES SEDELMEIER GOTTFRIED 2011-07-28 US disclosed
US-7943647-B2 Process for the preparation of tetrazole derivatives from organo aluminium azides NOVARTIS AG (CH) 2011-05-17 US disclosed
US-7943647-B2 Process for the preparation of tetrazole derivatives from organo aluminium azides NOVARTIS AG (CH) 2011-05-17 US disclosed
US-20070043098-A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides NOVARTIS PHARMACEUTICALS CORPORATION 2007-02-22 US disclosed
US-20070043098-A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides NOVARTIS PHARMACEUTICALS CORPORATION 2007-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043098-A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides ABL1, TBCA, TBC1D5 AGTR1 2005/4885
US-20250282779-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES DHPS, THPO, TNNI3 AGTR1 1015/4885
US-20120330026-A1 PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES ABL1, TBCA, TBC1D5 AGTR1 2005/4885
US-20220106314-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES DHPS, THPO, TNNI3 AGTR1 1015/4885
US-20110184187-A1 PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES ABL1, TBCA, TBC1D5 AGTR1 2005/4885
US-20220340569-A1 SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES DHPS, THPO, TNNI3 AGTR1 1015/4885
US-12616697-B2 Methods of treatment with myosin modulator MYH2, MYH14, MYH10 AGTR1 528/4885
US-20250325531-A1 TREATMENT OF SYSTOLIC DYSFUNCTION FABP3, TNNI3, TNNT2 AGTR1 173/4885
US-20250339395-A1 COMPOUNDS CONTAINING S-N-VALERYL-N-{[2'-(1H-TETRAZOLE-5-YL)-BIPHENYL-4-YL]-METHYL}-VALINE AND (2R,4S)-5-BIPHENYL-4-YL-4-(3-CARBOXY-PROPIONYLAMINO)-2-METHYL-PENTANOIC ACID ETHYL ESTER MOIETIES AND CATIONS MME, DNPEP, ANPEP AGTR1 8/4885
US-20250241903-A1 TREATMENT OF SYSTOLIC DYSFUNCTION FABP3, TNNI3, TNNT2 AGTR1 173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.