SCHEMBL12469600

SCHEMBL12469600

CCN1CCN(c2cc(-c3cccc(N)n3)ccn2)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KARS1 Q15046 5/20 0.45
PIK3C3 Q8NEB9 1/20 0.44
NOS3 P29474 3/20 0.43
NOS1 P29475 3/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
SMG1 Q96Q15 3/20 0.42
MTOR P42345 1/20 0.42
KIT P10721 4/20 0.42
FLT3 P36888 4/20 0.42
RAD52 P43351 1/20 0.42
NTRK1 P04629 2/20 0.41
SRC P12931 2/20 0.41
CDK1 P06493 1/20 0.41
CDK2 P24941 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
SLC2A1 P11166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902067 0.86 MTOR (0.54) KARS1SMG1MTORRAD52HRH3
SCHEMBL12469602 0.85 HRH4 (0.45) NOS3NOS1HTR1ADRD2HTR2A
SCHEMBL902015 0.81 ITGB2 (0.46) KARS1SMG1MTOR
SCHEMBL901638 0.80 PRKD3 (0.43) KARS1NOS3NOS1SMG1MTOR
SCHEMBL24322998 0.77 HRH3 (0.56) RAD52HRH3
SCHEMBL1704599 0.76 CKS1B (0.51) KIT
SCHEMBL4180910 0.76 GAA (0.51) HTR1ADRD2HTR2ARAD52HRH3
SCHEMBL6921614 0.74 CDK1 (0.43) KARS1PIK3C3SMG1RAD52CDK1
SCHEMBL15345047 0.71 DRD4 (0.50) DRD2RAD52HRH3
SCHEMBL23901371 0.71 MTOR (0.52) KARS1SMG1MTORRAD52HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed