SCHEMBL12469602

SCHEMBL12469602

CCN1CCN(c2cc(-c3cccc(N)n3)cc(N)n2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.45
NOS1 P29475 5/20 0.44
NOS3 P29474 4/20 0.44
HRH3 Q9Y5N1 1/20 0.43
KIT P10721 4/20 0.41
FLT3 P36888 4/20 0.41
DRD2 P14416 2/20 0.40
HTR2A P28223 2/20 0.40
HTR1A P08908 1/20 0.40
ASIC3 Q9UHC3 1/20 0.40
RAD52 P43351 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
GFER P55789 1/20 0.39
CYP2D6 P10635 2/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902069 0.85 HRH4 (0.57) HRH4HRH3
SCHEMBL12469600 0.85 KARS1 (0.45) NOS1NOS3HRH3KITFLT3
SCHEMBL24322998 0.82 HRH3 (0.56) HRH3RAD52SMN1; SMN2KDM4EGAA
SCHEMBL902018 0.80 NCF1 (0.52) HRH4NOS1NOS3GFERCNR2
SCHEMBL5452265 0.71 DRD2 (0.50) HRH3DRD2KDM4E
SCHEMBL902067 0.70 MTOR (0.54) HRH4HRH3RAD52KDM4E
SCHEMBL10112451 0.69 HRH3 (0.49) HRH3DRD2HTR2AHTR1ASMN1; SMN2
SCHEMBL3450414 0.68 HPGD (0.67) HRH4HRH3SMN1; SMN2KDM4EGAA
SCHEMBL3869622 0.68 HTR7 (0.47) HRH3DRD2SMN1; SMN2KDM4EMAPT
SCHEMBL22650478 0.67 CXCR4 (0.49) NOS1NOS3HRH3RAD52SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed