SCHEMBL12473602

SCHEMBL12473602

COc1ccc(CC(C=O)NC(=O)[C@@H](NC(=O)O)C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.50
CASP1 P29466 1/20 0.48
LDHA P00338 1/20 0.47
CTSD P07339 1/20 0.43
ACACB O00763 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12473613 0.87 CTSB (0.47) CTSBCASP1ACACB
SCHEMBL18262577 0.87 LDHA (0.57) CTSBLDHAACACBALDH1A1
SCHEMBL20204722 0.86 CTSB (0.62) CTSB
SCHEMBL12475011 0.85 CTSB (0.59) CTSBMMP9
SCHEMBL10084585 0.85 CTSB (0.62) CTSBCTSD
SCHEMBL7806376 0.85 CTSB (0.62) CTSBCTSD
SCHEMBL623793 0.85 ALDH1A1 (0.54) CTSBCASP1CTSDALDH1A1MMP3
SCHEMBL10084885 0.83 CASP1 (0.46) CTSBCASP1CTSDALDH1A1
SCHEMBL29537416 0.82 CTSD (0.50) CASP1CTSDMMP1MMP2MMP3
SCHEMBL622452 0.82 CASP1 (0.45) CTSBCASP1CTSDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed