SCHEMBL12474232

SCHEMBL12474232

N#Cc1ccc2nc(-c3ccc(-c4ccc(C5CC[CH]CC5)cc4)cc3)[nH]c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.58
PKN2 Q16513 1/20 0.58
CHEK2 O96017 2/20 0.55
DGAT1 O75907 6/20 0.53
KCNH2 Q12809 4/20 0.53
SOAT1 P35610 3/20 0.53
FASN P49327 3/20 0.49
RHEB Q15382 1/20 0.49
METAP2 P50579 1/20 0.46
METAP1 P53582 1/20 0.46
CSNK1A1 P48729 1/20 0.45
CSNK1D P48730 1/20 0.45
GSK3B P49841 1/20 0.45
CSNK1G2 P78368 1/20 0.45
SSTR2 P30874 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
RXFP1 Q9HBX9 2/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902210 0.89 PKN1 (0.60) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL20982510 0.82 PKN1 (0.82) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL901002 0.81 DGAT1 (0.74) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL3341423 0.76 PKN1 (0.72) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL14816640 0.76 PKN1 (0.72) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL18764054 0.76 CHEK2 (0.78) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL23563056 0.74 PKN1 (0.68) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL1662880 0.73 MEN1 (0.77) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL6061287 0.72 PKN1 (0.65) PKN1PKN2CHEK2DGAT1KCNH2
SCHEMBL7734383 0.72 GRIA1 (0.41) KCNH2NPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed