SCHEMBL12528005

SCHEMBL12528005

O=C(O)CC(CC(=O)O)(C(=O)O)C(O)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 3/20 0.58
CPT2 P23786 1/20 0.58
ALDH1A1 P00352 1/20 0.40
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
TDP1 Q9NUW8 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HMGCR P04035 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
ADRA1A P35348 1/20 0.35
TET2 Q6N021 3/20 0.32
KDM4A O75164 2/20 0.32
KDM4C Q9H3R0 2/20 0.32
KDM2A Q9Y2K7 2/20 0.32
TET3 O43151 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32
HSPD1 P10809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18798915 0.77 ACLY (0.43) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL12524010 0.77 ACLY (0.43) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL19258711 0.76 ALDH1A1 (0.46) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL9251690 0.75 CPT2 (0.41) ACLYCPT2ALDH1A1TSHRTDP1
SCHEMBL4951671 0.75 CPT2 (0.41) ACLYCPT2ALDH1A1TSHRTDP1
SCHEMBL721435 0.73 ACLY (1.00) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL17181757 0.73 ACLY (1.00) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL17181773 0.73 ACLY (1.00) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL6773065 0.73 ACLY (1.00) ACLYCPT2ALDH1A1CYP2D6TSHR
SCHEMBL2110910 0.73 ACLY (1.00) ACLYCPT2ALDH1A1CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170232013-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF MUSCULOSKELETAL RELATED DISEASES AND DISORDERS USING METAL ION-CITRATE ANALOG COMPLEXES THE CHARLOTTE-MECKLENBURG HOSPITAL AUTHORITY D/B/A ATRIUM HEALTH 2017-08-17 US disclosed
US-9636352-B2 Compositions and methods for the treatment of musculoskeletal related diseases and disorders using metal ion-citrate analog complexes THE CHARLOTTE-MECKLENBURG HOSPITAL AUTHORITY (US) 2017-05-02 US disclosed
WO-2012125524-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF MUSCULOSKELETAL RELATED DISEASES AND DISORDERS USING METAL ION-CITRATE ANALOG COMPLEXES THE CHARLOTTE-MECKLENBURG HOSPITAL AUTHORITY D/B/A CAROLINAS MEDICAL CENTER (US) 2012-09-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170232013-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF MUSCULOSKELETAL RELATED DISEASES AND DISORDERS USING METAL ION-CITRATE ANALOG COMPLEXES CS, ACLY, CA5A ACLY 2/4885CPT2 288/4885ALDH1A1 1294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.