SCHEMBL1266601

SCHEMBL1266601

COc1nc(Cl)ccc1C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MERTK Q12866 1/20 0.43
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
ALDH1A1 P00352 8/20 0.39
NFE2L2 Q16236 1/20 0.38
GAA P10253 3/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TRIM24 O15164 1/20 0.38
TYR P14679 1/20 0.38
TRIM33 Q9UPN9 1/20 0.38
LMNA P02545 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ERN1 O75460 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392617 1.00 MERTK (0.43) MERTKCRHBPCRHR2ALDH1A1NFE2L2
SCHEMBL30023734 0.81 NCF1 (0.44) ALDH1A1GAATRIM24TYRTRIM33
SCHEMBL17559335 0.80 ALDH1A1 (0.56) CRHBPCRHR2ALDH1A1GAAHPGD
SCHEMBL9831052 0.80 ALDH1A1 (0.41) ALDH1A1GAASMN1; SMN2TRIM24TYR
SCHEMBL29952654 0.78 ERN1 (0.52) ALDH1A1HPGDSMN1; SMN2TRIM24TYR
SCHEMBL1534756 0.78 ERN1 (0.52) ALDH1A1HPGDSMN1; SMN2TRIM24TYR
SCHEMBL30433024 0.77 PDCD1LG2 (0.58)
SCHEMBL21497019 0.77 PDCD1LG2 (0.58)
SCHEMBL2415421 0.77 PRKDC (0.40) ALDH1A1GAATRIM24TYRTRIM33
SCHEMBL30772448 0.77 ALDH1A1 (0.39) ALDH1A1GAATRIM24TYRTRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 378 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118702774-A Preparation method and application of polypeptide coupling compound of targeted GPC-3 protein 上海大学 2024-09-27 CN claimed
CN-117683021-A PD-1/PD-L1 pathway targeting compound and nuclide marker, preparation and application thereof 厦门大学 2024-03-12 CN claimed
EP-4746972-A1 DEUTERATED PARP1 INHIBITOR COMPOUNDS Duke Street Bio Limited (GB) 2026-05-27 EP disclosed
CN-122079995-A PD-1/PD-L1 and JAK double-target inhibitor, preparation method and application 2026-05-26 CN disclosed
EP-4234030-B1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES INC (US) 2026-04-08 EP disclosed
US-12590062-B2 PD-1/PD-L1 inhibitors GILEAD SCIENCES, INC. (US) 2026-03-31 US disclosed
US-12583822-B2 Benzylamine derivative, preparation method therefor and use thereof ACADEMY OF MILITARY MEDICAL SCIENCES (CN) 2026-03-24 US disclosed
EP-4045036-B1 HETEROARYL-BIPHENYL AMIDES FOR THE TREATMENT OF PD-L1 DISEASES CHEMOCENTRYX INC (US) 2026-03-04 EP disclosed
US-20260042779-A1 SYNTHESIS OF SUBSTITUTED 1-ARYL-1'-HETEROARYL COMPOUNDS AND SUBSTITUTED 1,1'-BIHETEROARYL COMPOUNDS, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORPORATION (CA) 2026-02-12 US disclosed
EP-4045037-B1 HETEROARYL-BIPHENYL AMINES FOR THE TREATMENT OF PD-L1 DISEASES CHEMOCENTRYX INC (US) 2026-01-28 EP disclosed
EP-4680226-A2 ACYLSULFONAMIDE KAT6A INHIBITORS Olema Pharmaceuticals, Inc. (US) 2026-01-21 EP disclosed
EP-0565621-A1 METHOD OF MAKING CAMPTOTHECIN AND CAMPTOTHECIN ANALOGS NORTH CAROLINA STATE UNIVERSITY (US) 1993-10-20 EP disclosed
US-5254690-A Alkoxymethylpyridine d-ring intermediates useful for the synthesis of camptpthecin and camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1993-10-19 US disclosed
US-5247089-A Method of making intermediates useful for the manufacture of camptothecin and camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1993-09-21 US disclosed
US-5243050-A Alkylpyridone DE ring intermediates useful for the manufacture of camptothecin and camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1993-09-07 US disclosed
US-5212317-A Methods and intermediates for the assymmetric synthesis of camptothecin and camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1993-05-18 US disclosed
US-5200524-A Camptothecin intermediates and method of making same NORTH CAROLINA STATE UNIVERSITY (US) 1993-04-06 US disclosed
US-5191082-A Camptothecin intermediate and method of making camptothecin intermediates NORTH CAROLINA STATE UNIVERSITY (US) 1993-03-02 US disclosed
US-5162532-A INTERMEDIATES AND METHOD OF MAKING CAMPTOTHECIN AND CAMPTOTHECIN ANALOGS NORTH CAROLINA STATE UNIVERSITY (US) 1992-11-10 US disclosed
WO-1992011263-A1 METHOD OF MAKING CAMPTOTHECIN AND CAMPTOTHECIN ANALOGS NORTH CAROLINA STATE UNIVERSITY (US) 1992-07-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260042779-A1 SYNTHESIS OF SUBSTITUTED 1-ARYL-1'-HETEROARYL COMPOUNDS AND SUBSTITUTED 1,1'-BIHETEROARYL COMPOUNDS, AND ANALOGUES THEREOF HAVCR2, NNMT, DOHH MERTK 4085/4885CRHBP 4406/4885CRHR2 4231/4885
US-12583822-B2 Benzylamine derivative, preparation method therefor and use thereof CD274, PDCD1, PDCD1LG2 MERTK 4545/4885CRHBP 1800/4885CRHR2 317/4885
US-12590062-B2 PD-1/PD-L1 inhibitors CD274, PDCD1LG2, PDCD1 MERTK 3273/4885CRHBP 2922/4885CRHR2 571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.