SCHEMBL1273290

SCHEMBL1273290

C[C@@H]1OC[C@@H](c2ccccc2)N(C(=O)OC(C)(C)C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 6/20 0.42
RORC P51449 2/20 0.39
ABCB1 P08183 1/20 0.39
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
GPR119 Q8TDV5 1/20 0.38
KLK7 P49862 1/20 0.38
ACHE P22303 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1274642 0.84 RIPK1 (0.45) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL1274450 0.83 ALDH1A1 (0.40) RIPK1
SCHEMBL1274502 0.79 RIPK1 (0.46) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL12901410 0.78 USP2 (0.36) NR1H2
SCHEMBL248353 0.78 RIPK1 (0.61) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL10061592 0.78 RIPK1 (0.61) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL15850701 0.78 RIPK1 (0.61) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL1274811 0.75 RIPK1 (0.45) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL18448056 0.74 RIPK1 (0.49) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL7589379 0.74 L3MBTL1 (0.51) RIPK1RORCABCB1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7893079-B2 Substituted monocyclic CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-02-22 US disclosed