SCHEMBL1274502

SCHEMBL1274502

CC(C)(C)OC(=O)N1C(=O)COC[C@H]1c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 5/20 0.46
RORC P51449 2/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ABCB1 P08183 1/20 0.39
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
GPR119 Q8TDV5 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KLK7 P49862 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL248353 0.85 RIPK1 (0.61) RIPK1RORCHDAC1HDAC8HDAC6
SCHEMBL10061592 0.85 RIPK1 (0.61) RIPK1RORCHDAC1HDAC8HDAC6
SCHEMBL15850701 0.85 RIPK1 (0.61) RIPK1RORCHDAC1HDAC8HDAC6
SCHEMBL1274378 0.82 RIPK1 (0.38) RIPK1HDAC1HDAC8HDAC6
SCHEMBL1274529 0.81 ALDH1A1 (0.42) RIPK1HDAC1HDAC8HDAC6
SCHEMBL7589379 0.80 L3MBTL1 (0.51) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL1273290 0.79 RIPK1 (0.42) RIPK1RORCHDAC1HDAC8HDAC6
SCHEMBL20879577 0.77 NR1H2 (0.46) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL29695962 0.77 MDM2 (0.42) RIPK1RORCABCB1NR1H2NR1H3
SCHEMBL23522781 0.76 USP2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7893079-B2 Substituted monocyclic CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-02-22 US disclosed