SCHEMBL12765737

SCHEMBL12765737

c1ccc2c(CC3CC3)c[nH]c2c1

nearest known ligand 0.81

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.81
HTR6 P50406 8/20 0.64
KMT2A Q03164 3/20 0.62
MAPT P10636 2/20 0.62
MEN1 O00255 1/20 0.62
CYP3A4 P08684 1/20 0.62
AHR P35869 1/20 0.62
GPR84 Q9NQS5 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
POLB P06746 1/20 0.56
HPGD P15428 1/20 0.56
BCHE P06276 1/20 0.56
CYP2D6 P10635 1/20 0.56
LMNA P02545 2/20 0.55
HTT P42858 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL733304 0.91 SLC6A4 (0.73) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL1998835 0.90 SLC6A4 (1.00) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL30592374 0.90 SLC6A4 (1.00) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL4822564 0.85 SLC6A4 (0.71) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL27923059 0.83 SLC6A4 (0.82) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL14282331 0.83 HTR1A (0.65) SLC6A4HTR6BCHECYP2D6
SCHEMBL24178316 0.81 HTR6 (0.69) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL30361714 0.81 HTR6 (0.69) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL24178288 0.81 HTR6 (0.69) SLC6A4HTR6KMT2AMAPTMEN1
SCHEMBL31302667 0.81 SLC6A4 (0.68) SLC6A4HTR6KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11873305-B2 Processes for synthesis of substituted indole intermediates for the synthesis of serd compounds GENENTECH, INC. (US) 2024-01-16 US disclosed
CN-108101830-B A kind of 3- replaces the preparation method of Oxoindole and derivative 中国科学院成都生物研究所 2019-08-23 CN disclosed
US-7897619-B2 Heterocyclic modulators of PKB AMGEN INC. (US) 2011-03-01 US disclosed
US-20090275592-A1 Heterocyclic modulators of PKB AMGEN INC. (US) 2009-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11873305-B2 Processes for synthesis of substituted indole intermediates for the synthesis of serd compounds WEE1, WEE2, INMT SLC6A4 626/4885HTR6 425/4885KMT2A 2114/4885
US-20090275592-A1 Heterocyclic modulators of PKB MTOR, PDK1, EIF4EBP1 SLC6A4 4618/4885HTR6 1758/4885KMT2A 3140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.