SCHEMBL12877478

SCHEMBL12877478

C=CC[C@H](NC(=O)c1ccccc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.50
ACE P12821 2/20 0.49
PIN1 Q13526 1/20 0.49
CYP2C19 P33261 1/20 0.49
PTPN1 P18031 2/20 0.48
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
CTSL P07711 1/20 0.47
CTRB1 P17538 1/20 0.46
SLC1A2 P43004 1/20 0.46
IDO1 P14902 1/20 0.46
CA2 P00918 4/20 0.46
CA1 P00915 2/20 0.46
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL712558 1.00 FOLH1 (0.50) FOLH1ACEPIN1CYP2C19PTPN1
SCHEMBL5727358 0.87 ALDH1A1 (0.46) CYP2C19ALDH1A1LMNAHPGDCTSL
SCHEMBL714529 0.84 TAS1R3 (0.54) ALDH1A1LMNACTSL
SCHEMBL8232716 0.84 TAS1R3 (0.54) ALDH1A1LMNACTSL
SCHEMBL2782642 0.84 TAS1R3 (0.54) ALDH1A1LMNACTSL
SCHEMBL3187487 0.84 POLB (0.49) FOLH1PIN1CYP2C19ALDH1A1LMNA
SCHEMBL5761847 0.82 PKM (0.57) FOLH1PTPN1ALDH1A1LMNACTSL
SCHEMBL714183 0.81 CA2 (0.57) FOLH1ALDH1A1LMNACA2CA1
SCHEMBL11063949 0.81 ACE (0.52) ACEPTPN1ALDH1A1CTSLSLC1A2
SCHEMBL713931 0.81 ICMT (0.47) ACEPIN1CYP2C19PTPN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984384-B1 Conotoxin analogues, and methods for synthesis of intramolecular dicarba bridge containing peptides SYNGENE LTD (AU) 2015-10-21 EP disclosed
WO-2011015241-A1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2011-02-10 WO disclosed