SCHEMBL13061114

SCHEMBL13061114

CCc1cccc(-c2cccc(C(=O)N[C@H](CN(C)C)C(C)C)c2)c1OC

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 3/20 0.41
TAS1R1 Q7RTX1 3/20 0.41
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
UTS2R Q9UKP6 6/20 0.39
HDAC4 P56524 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060800 1.00 TAS1R3 (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13005536 0.92 ROCK2 (0.40) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13005534 0.92 ROCK2 (0.40) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060890 0.86 CTSL (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060892 0.86 CTSL (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13061023 0.84 ROCK2 (0.51) ROCK2ROCK1UTS2R
SCHEMBL13060640 0.83 TAS1R3 (0.40) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060643 0.82 ROCK2 (0.44) ROCK2ROCK1HDAC4
SCHEMBL13061226 0.82 ROCK2 (0.44) ROCK2ROCK1HDAC4
SCHEMBL13060641 0.81 MEN1 (0.41) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed