SCHEMBL13071404

SCHEMBL13071404

CCOC(=O)[C@H]1C[C@H]1/C=C\CCCCC[C@H](Nc1cccc(C(F)(F)F)c1)C(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HSP90AA1 P07900 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
GAA P10253 3/20 0.35
MAPT P10636 1/20 0.35
ATM Q13315 1/20 0.35
CCR1 P32246 1/20 0.35
XIAP P98170 2/20 0.34
DPP4 P27487 2/20 0.34
ACE P12821 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071527 0.92 DPP4 (0.39) ALDH1A1SMN1; SMN2CCR1XIAPDPP4
SCHEMBL13072076 0.91 ACE (0.35) ALDH1A1SMN1; SMN2GAAACELMNA
SCHEMBL13071880 0.91 UBE2M (0.34) ALDH1A1SMN1; SMN2XIAPDPP4ACE
SCHEMBL12831754 0.90 ACE (0.41) SMN1; SMN2ACELMNA
SCHEMBL13071526 0.89 UBE2M (0.35) XIAPACEUBE2MDCUN1D1
SCHEMBL13071528 0.87 DPP4 (0.36) SMN1; SMN2DPP4ACELMNA
SCHEMBL13071885 0.86 XIAP (0.35) SMN1; SMN2GAAMAPTCCR1XIAP
SCHEMBL13071388 0.83 HTR1A (0.38) ALDH1A1SMN1; SMN2MAPTACELMNA
SCHEMBL13071921 0.81 DPP4 (0.35) XIAPDPP4ACEUBE2MDCUN1D1
SCHEMBL8203250 0.79 F2 (0.41) ACECTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed