SCHEMBL13075508

SCHEMBL13075508

Nc1cnc(-c2c(Cl)cccc2C(F)(F)F)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.41
PTGES O14684 3/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABL1 P00519 1/20 0.36
TRPA1 O75762 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
MAPK14 Q16539 1/20 0.34
MPL P40238 1/20 0.34
NPY5R Q15761 1/20 0.34
SCN9A Q15858 2/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AXL P30530 1/20 0.33
HRH1 P35367 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
PIK3CD O00329 1/20 0.33
SCN2A Q99250 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13075496 0.84 JAK2 (0.54) JAK2PTGESHRH1SCN2A
SCHEMBL3797673 0.84 JAK2 (0.42) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL3799817 0.79 PDE4A (0.39) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL13075509 0.74 PTGES (0.43) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL30962796 0.70 ABL1 (0.42) ABL1SCN9APPARGRORC
SCHEMBL3795873 0.69 PTGES (0.49) JAK2PTGES
SCHEMBL3798446 0.67 TRPA1 (0.44) PTGESTRPA1NPY5RSCN9AALDH1A1
SCHEMBL15401823 0.66 ABL1 (0.60) JAK2ABL1TRPA1PIK3CD
SCHEMBL3800300 0.66 PTGES (0.43) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL31571903 0.66 P2RX7 (0.40) MAPK14MPLALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed