SCHEMBL3797673

SCHEMBL3797673

FC(F)(F)c1cnc(-c2c(Cl)cccc2C(F)(F)F)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.42
PTGES O14684 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
DGAT1 O75907 2/20 0.38
RAF1 P04049 4/20 0.37
ABL1 P00519 1/20 0.37
AURKA O14965 2/20 0.36
KDR P35968 2/20 0.36
ERBB2 P04626 1/20 0.36
TRPA1 O75762 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
NPY5R Q15761 1/20 0.35
AXL P30530 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3795873 0.85 PTGES (0.49) JAK2PTGESDGAT1
SCHEMBL13075508 0.84 JAK2 (0.41) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL3798446 0.83 TRPA1 (0.44) PTGESDGAT1AURKAKDRERBB2
SCHEMBL3799817 0.80 PDE4A (0.39) JAK2PTGESCYP3A4CYP2C9CYP2C19
SCHEMBL25754915 0.76 DGAT1 (0.41) PTGESDGAT1AURKAKDRERBB2
SCHEMBL23847031 0.71 TSHR (0.41) DGAT1AURKAKDRERBB2SMN1; SMN2
SCHEMBL11245211 0.71 HRH1 (0.56) NPY5RKDM4EALDH1A1
SCHEMBL30077144 0.71 AURKA (0.39) DGAT1RAF1AURKAKDRERBB2
SCHEMBL15347521 0.71 AURKA (0.39) DGAT1RAF1AURKAKDRERBB2
SCHEMBL13075509 0.70 PTGES (0.43) JAK2PTGESCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed