SCHEMBL13076381

SCHEMBL13076381

Fc1ccc(C2(c3nc(-c4ccc(-c5c[nH]c(-c6c(F)cccc6Cl)n5)cn4)no3)CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.34
NPC1 O15118 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PTGES O14684 5/20 0.33
CHRNB2 P17787 4/20 0.32
CHRNA4 P43681 4/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
REN P00797 1/20 0.31
CYP3A4 P08684 1/20 0.31
KCNH2 Q12809 1/20 0.31
MAPK9 P45984 1/20 0.31
MAPK10 P53779 1/20 0.31
MAPK11 Q15759 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3799989 0.87 PTGES (0.44) HSD11B1NPC1CASP3RAB9ASENP8
SCHEMBL13076233 0.80 RAB9A (0.43) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL13076261 0.79 GRM5 (0.41) HSD11B1NPC1RAB9APTGESCHRNB2
SCHEMBL13076379 0.79 GRM5 (0.45) HSD11B1NPC1RAB9ACHRNB2CHRNA4
SCHEMBL13076382 0.78 HTT (0.42) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL13076244 0.78 NPC1 (0.43) HSD11B1NPC1CASP3RAB9ASENP7
SCHEMBL13076236 0.77 NPC1 (0.45) HSD11B1NPC1CASP3RAB9ASENP7
SCHEMBL13076380 0.76 PTGES (0.35) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL13076263 0.76 NPC1 (0.35) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL13076262 0.76 RAB9A (0.45) NPC1CASP3RAB9ASENP8SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed