SCHEMBL13176993

SCHEMBL13176993

Cc1c(Cl)cccc1Nc1nc2ccc(S(=O)(=O)Cc3ccccc3)c(C(=O)O)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 17/20 0.42
MT-CO2 P00403 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
TTR P02766 1/20 0.41
PLA2G1B P04054 1/20 0.41
CYP1A2 P05177 1/20 0.41
PGR P06401 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
AR P10275 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
HTR2A P28223 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927954 0.91 MAPT (0.39) P2RX7MAPTKMT2A
SCHEMBL13989967 0.89 P2RX7 (0.42) P2RX7MEN1MAPTKMT2A
SCHEMBL2925195 0.84 NPC1 (0.40) P2RX7MAPTKMT2A
SCHEMBL2932570 0.78 MAPT (0.42) MEN1LMNAMAPTKMT2A
SCHEMBL13989934 0.76 MEN1 (0.45) MEN1LMNAMAPTKMT2A
SCHEMBL14628462 0.75 CA2 (0.37) MEN1LMNAKMT2A
SCHEMBL2925046 0.71 MAPT (0.39) P2RX7MEN1LMNAARMAPT
SCHEMBL13176992 0.70 LMNA (0.38) LMNAARMAPTHIF1A
SCHEMBL2931581 0.69 POLB (0.55) MT-CO2MEN1USP2LMNATTR
SCHEMBL1115893 0.69 MAPT (0.42) MEN1LMNAMAPTKMT2ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910314-B1 BENZIMIDAZOLE DERIVATIVES FOR TREATMENT OF INFLAMMATORY DISEASES NOVARTIS AG (CH) 2010-09-15 EP disclosed