SCHEMBL133151

SCHEMBL133151

C(=C/c1ccc(N(c2ccccc2)c2ccccc2)cc1)\c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 3/20 0.64
ALDH1A1 P00352 3/20 0.52
MAOB P27338 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
MAPT P10636 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
NFE2L2 Q16236 1/20 0.52
CYP19A1 P11511 1/20 0.52
MAOA P21397 1/20 0.52
APP P05067 1/20 0.50
CTDSP1 Q9GZU7 1/20 0.47
TRPA1 O75762 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.45
MEN1 O00255 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13720653 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL14005735 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL9971916 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL10128952 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL243730 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL13720595 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL13136849 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL243731 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL133152 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E
SCHEMBL5338475 1.00 RELA (0.64) RELAALDH1A1MAOBL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 162 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4596754-A Electroconductive support, photosensitive layer comprising azo pigment charge generating layer, charge transport layer, alkali soluble resin RICOH COMPANY, LTD. (JP) 1986-06-24 US claimed
US-20240373749-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT KYULUX, INC. (JP) 2024-11-07 US disclosed
US-12089494-B2 Organic electroluminescence element KYUSHU UNIVERSITY, NATIONAL UNIVERSITY CORPORATION (JP) 2024-09-10 US disclosed
US-11287756-B2 Positive charging electrophotographic photoreceptor, electrophotographic cartridge and image forming apparatus MITSUBISHI CHEMICAL CORPORATION (JP) 2022-03-29 US disclosed
US-20210387994-A1 SOLVENT-FREE CROSS-COUPLING REACTION, AND PRODUCTION METHOD USING SAID REACTION NATIONAL UNIVERSITY CORPORATION HOKKAIDO UNIVERSITY (JP) 2021-12-16 US disclosed
US-20210202864-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT KYULUX, INC. (JP) 2021-07-01 US disclosed
EP-3843167-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT Kyushu University, National University Corporation (JP) 2021-06-30 EP disclosed
US-10761439-B2 Polyarylate resin and electrophotographic photosensitive member KYOCERA DOCUMENT SOLUTIONS INC. (JP) 2020-09-01 US disclosed
US-10651390-B2 Tertiary amine compound, photoelectric conversion element, and solar cell RICOH COMPANY, LTD. (JP) 2020-05-12 US disclosed
WO-2020085396-A1 SOLVENT-FREE CROSS-COUPLING REACTION, AND PRODUCTION METHOD USING SAID REACTION 国立大学法人北海道大学 2020-04-30 WO disclosed
US-4716220-A CHARGE CARRIER GENERATING MATERIALS RICOH CO., LTD. (JP) 1987-12-29 US disclosed
US-4708921-A Photosensitive material containing disazo compound for use in electrophotography RICOH CO., LTD. (JP) 1987-11-24 US disclosed
US-4702979-A ELECTROCONDUCTIVE CATHODE LAYER, PHOTOCONDUCTIVE LAYER OF CHARGE-GENERATING ORGANIC PIGMENT, ANODIC ION REACTION AT INTERFACE WHEN IRRADIATED RICOH CO., LTD. (JP) 1987-10-27 US disclosed
US-4672149-A PHOTOACTIVE LAYER CONTAINING A DISAZO PIGMENT; SOLAR CELLS; EFFICIENCY RICOH CO., LTD. (JP) 1987-06-09 US disclosed
US-4663442-A ELECTROGRAPHY, PHOTOSENSITIVITY RICOH CO., LTD. (JP) 1987-05-05 US disclosed
US-4619878-A Tetrazonium salt compound, disazo compound, method for preparing the same, and photosensitive material containing said disazo compound for use in electrophotography RICOH CO., LTD. (JP) 1986-10-28 US disclosed
US-4596754-A Electroconductive support, photosensitive layer comprising azo pigment charge generating layer, charge transport layer, alkali soluble resin RICOH COMPANY, LTD. (JP) 1986-06-24 US disclosed
US-4582771-A Disazo compound, method for preparing the same, and electrophotographic element containing the same for use in electrophotography RICOH CO., LTD. (JP) 1986-04-15 US disclosed
US-4565759-A PHOTOCONDUCTIVE LAYER ON ELECTROCONDUCTIVE SUPPORT RICOH CO., LTD. (JP) 1986-01-21 US disclosed
US-4540643-A Tetrazonium salt compounds, novel disazo compounds, method for the production thereof and disazo compound-containing electrophotographic elements RICOH CO., LTD. (JP) 1985-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240373749-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT LEF1, EMC1, EEA1 RELA 1945/4885ALDH1A1 157/4885MAOB 2896/4885
US-12089494-B2 Organic electroluminescence element LEF1, EMC1, EEA1 RELA 1945/4885ALDH1A1 157/4885MAOB 2896/4885
US-20210387994-A1 SOLVENT-FREE CROSS-COUPLING REACTION, AND PRODUCTION METHOD USING SAID REACTION MCCC2, CTRC, DDC RELA 1869/4885ALDH1A1 2438/4885MAOB 108/4885
US-10651390-B2 Tertiary amine compound, photoelectric conversion element, and solar cell SUN2, CRY1, TEAD1 RELA 2496/4885ALDH1A1 631/4885MAOB 2093/4885
US-20210202864-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT LEF1, EMC1, EEA1 RELA 1945/4885ALDH1A1 157/4885MAOB 2896/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.