SCHEMBL1343400

SCHEMBL1343400

CC1C(=O)NCCN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
PARP1 P09874 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
DDB1 Q16531 2/20 0.38
CRBN Q96SW2 2/20 0.38
DPP4 P27487 1/20 0.37
ALDH1A1 P00352 1/20 0.37
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.35
GPR119 Q8TDV5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19474636 1.00 MAPK1 (0.41) MAPK1PARP1L3MBTL1KDM4EMAPT
SCHEMBL14850713 1.00 MAPK1 (0.41) MAPK1PARP1L3MBTL1KDM4EMAPT
SCHEMBL3995391 0.91 DPP4 (0.43) PARP1DPP4HSD17B10
SCHEMBL7341850 0.90 DPP4 (0.42) PARP1DPP4HSD17B10
SCHEMBL17596640 0.84 MAPK1 (0.41) MAPK1PARP1KDM4EMAPTTHRB
SCHEMBL17596585 0.84 MAPK1 (0.41) MAPK1PARP1KDM4EMAPTTHRB
SCHEMBL1343753 0.81 L3MBTL1 (0.44) MAPK1PARP1L3MBTL1KDM4EMAPT
SCHEMBL15271978 0.81 MAPK1 (0.39) MAPK1PARP1L3MBTL1KDM4EMAPT
SCHEMBL2674093 0.81 MAPK1 (0.39) MAPK1PARP1L3MBTL1KDM4EMAPT
SCHEMBL13223548 0.79 DPP4 (0.39) L3MBTL1KDM4EDPP4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119462531-A Preparation of non-azole Process for preparing tam intermediates 广东莱佛士制药技术有限公司 2025-02-18 CN claimed
US-12565500-B2 Substituted pyrrolo[1,2-b]pyridazines and pyrrolo[2,1-f][1,2,4]triazines as Btk inhibitors BIOGEN MA INC. (US) 2026-03-03 US disclosed
EP-4658262-A1 BICYCLIC IMIDE COMPOUNDS AS TRPA1 INHIBITORS D.E. Shaw Research, LLC (US) 2025-12-10 EP disclosed
EP-4638455-A1 HETEROCYCLIC GLP-1 AGONISTS Gasherbrum Bio, Inc. (US) 2025-10-29 EP disclosed
EP-4051679-B1 CONDENSED PYRIDAZINE OR PYRIMIDINE AS BTK INHIBITORS BIOGEN MA INC (US) 2025-08-06 EP disclosed
US-12338243-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2025-06-24 US disclosed
CN-119462531-A Preparation of non-azole Process for preparing tam intermediates 广东莱佛士制药技术有限公司 2025-02-18 CN disclosed
CN-119462531-A Preparation of non-azole Process for preparing tam intermediates 广东莱佛士制药技术有限公司 2025-02-18 CN disclosed
US-20250034150-A1 BTK INHIBITORS BIOGEN MA INC. 2025-01-30 US disclosed
CN-118804915-A BTK inhibitors 渤健马萨诸塞州股份有限公司 2024-10-18 CN disclosed
US-20140275097-A1 NOVEL CHIRAL N-ACYL-5,6,7(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF OGEDA SA (BE) 2014-09-18 US disclosed
WO-2013050424-A1 NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF EUROSCREEN S.A. (BE) 2013-04-11 WO disclosed
US-8063042-B2 Heterocyclic compounds HOFFMANN-LA ROCHE INC. (US) 2011-11-22 US disclosed
US-8044069-B2 Compounds as calcium channel blockers ABBOTT LABORATORIES (US) 2011-10-25 US disclosed
EP-2307387-A1 NOVEL HETEROCYCLYL COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISEASE F. Hoffmann-La Roche AG (CH) 2011-04-13 EP disclosed
WO-2011041713-A2 PIPERAZINYL ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-07 WO disclosed
EP-2220055-A2 NOVEL HETEROCYCLYL COMPOUNDS AND THEIR USE AS CHEMOKINE ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2010-08-25 EP disclosed
US-20100093730-A1 NOVEL COMPOUNDS AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-04-15 US disclosed
US-20090023713-A1 HETEROCYCLIC COMPOUNDS HOFFMANN-LA ROCHE, INC. 2009-01-22 US disclosed
WO-2009010429-A2 NOVEL HETEROCYCLYL COMPOUNDS AND THEIR USE AS CHEMOKINE ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-01-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093730-A1 NOVEL COMPOUNDS AS CALCIUM CHANNEL BLOCKERS CACNA1E, CACNA1S, CACNA1D MAPK1 1458/4885PARP1 2280/4885L3MBTL1 1998/4885
US-12338243-B2 P2X7 modulators P2RX7, P2RX4, P2RX1 MAPK1 937/4885PARP1 2653/4885L3MBTL1 4865/4885
US-20140275097-A1 NOVEL CHIRAL N-ACYL-5,6,7(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF ACKR3, GPR3, TAC3 MAPK1 3623/4885PARP1 1945/4885L3MBTL1 4750/4885
US-20090023713-A1 HETEROCYCLIC COMPOUNDS CCR5, CCR3, CCR2 MAPK1 1052/4885PARP1 1841/4885L3MBTL1 3686/4885
US-20250034150-A1 BTK INHIBITORS BTK, SYK, LYN MAPK1 293/4885PARP1 1629/4885L3MBTL1 3141/4885
US-12565500-B2 Substituted pyrrolo[1,2-b]pyridazines and pyrrolo[2,1-f][1,2,4]triazines as Btk inhibitors BTK, SYK, OXSR1 MAPK1 205/4885PARP1 662/4885L3MBTL1 3795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.