SCHEMBL1344836

SCHEMBL1344836

COC(=O)C(C)c1ccccc1Oc1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.46
CXCL8 P10145 3/20 0.44
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR2A P28223 2/20 0.40
SLC6A4 P31645 2/20 0.40
KCNH2 Q12809 1/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 1/20 0.39
CAMK2A Q9UQM7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11833301 0.84 CXCL8 (0.52) XIAPCXCL8ALDH1A1MAPTMEN1
SCHEMBL1346100 0.84 CXCL8 (0.52) XIAPCXCL8ALDH1A1MAPTMEN1
SCHEMBL13403891 0.84 CXCL8 (0.46) CXCL8ALDH1A1KMT2AHTR2ASLC6A4
SCHEMBL5706168 0.84 CXCL8 (0.46) CXCL8ALDH1A1KMT2AHTR2ASLC6A4
SCHEMBL31612955 0.84 CXCL8 (0.46) CXCL8ALDH1A1KMT2AHTR2ASLC6A4
SCHEMBL5541713 0.82 LPAR1 (0.49) ALDH1A1POLBKMT2AHPGD
SCHEMBL10937637 0.81 LMNA (0.51) MAPTMEN1POLBKMT2AHTR2A
SCHEMBL27423648 0.77 P2RX3 (0.37) ALDH1A1MAPTHTR2ASLC6A4KCNH2
SCHEMBL11435322 0.77 P2RX3 (0.49) XIAPCXCL8ALDH1A1HTR2ASLC6A4
Hydrochloric Acid SCHEMBL21494480 0.75 L3MBTL1 (0.49) ALDH1A1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229942-B1 2-Aryl-propionic acids and pharmaceutical compositions containing them DOMPE SPA (IT) 2012-08-29 EP disclosed
US-8063242-B2 for treatment of neutrofil-dependent pathologies such as psoriasis, ulcerative colitis, melanoma, chronic obstructive pulmonary disease (COPD), bollous pemphigo, rheumatoid arthritis, idiopathic fibrosis, glomerulonephritis; prevention and treatment of damages caused by ischemia and reperfusion DOMPE PHA.R.MA S.P.A. (IT) 2011-11-22 US disclosed
EP-2229942-A1 2-Aryl-propionic acids and pharmaceutical compositions containing them Dompe S.p.A. (IT) 2010-09-22 EP disclosed
US-20050038119-A1 2-Aryl-propionic acids and pharmaceutical compositions containing them DOMPÉ FARMACEUTICI S.P.A. (IT) 2005-02-17 US disclosed
EP-1455773-A1 2-ARYL-PROPIONIC ACIDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dompé S.P.A. (IT) 2004-09-15 EP disclosed
WO-2003043625-A1 2-ARYL-PROPIONIC ACIDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPE S.P.A. (IT) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038119-A1 2-Aryl-propionic acids and pharmaceutical compositions containing them CXCR2, FPR1, CCR2 XIAP 561/4885CXCL8 16/4885ALDH1A1 691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.