SCHEMBL13489152

SCHEMBL13489152

CN1c2ccccc2C(Cc2ccccc2)c2ccccc2N(C)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.49
CES2 O00748 1/20 0.44
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
ACHE P22303 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
HRH1 P35367 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5667766 0.98 EGFR (0.50) EGFRCES2HDAC4HDAC7HDAC5
SCHEMBL31613810 0.98 EGFR (0.50) EGFRCES2HDAC4HDAC7HDAC5
SCHEMBL3085394 0.76 EGFR (0.41) EGFRCES2HDAC4HDAC7HDAC5
SCHEMBL11537019 0.75 LTA4H (0.47) MEN1KMT2AKDM4C
SCHEMBL6997095 0.75 HTR2A (0.54) EGFRHDAC4HDAC7HDAC5ACHE
SCHEMBL8811499 0.74 EGFR (0.78) EGFRHDAC4HDAC7HDAC5ACHE
SCHEMBL3091840 0.74 EGFR (0.40) EGFRHDAC4HDAC7HDAC5ACHE
SCHEMBL9719345 0.73 ROCK2 (0.51) EGFRCES2MEN1KMT2AKDM4C
SCHEMBL3918548 0.71 HTR2A (0.54) MEN1KMT2AHTR2AEP300
SCHEMBL3797401 0.71 HDAC4 (0.52) EGFRHDAC4HDAC7HDAC5ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100041880-A1 Supramolecular Scaffolds and Methods of Making the Same LOYOLA UNIVERSITY OF CHICAGO (US) 2010-02-18 US disclosed
US-20100041880-A1 Supramolecular Scaffolds and Methods of Making the Same LOYOLA UNIVERSITY OF CHICAGO (US) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041880-A1 Supramolecular Scaffolds and Methods of Making the Same BLM, TBXAS1, TOP2B EGFR 3719/4885CES2 2310/4885HDAC4 3945/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.