SCHEMBL13508399

SCHEMBL13508399

C(=C(c1ccccc1)c1ccccc1)c1ccc(N(c2ccc(C=C(c3ccccc3)c3ccccc3)cc2)c2ccc(/C=C(\c3ccc4ccccc4c3)c3cccc4ccccc34)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.36
CYP2D6 P10635 2/20 0.36
PLAU P00749 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS2 P35354 2/20 0.36
CYP19A1 P11511 1/20 0.35
CYP11B2 P19099 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
F7 P08709 1/20 0.35
AKR1C2 P52895 1/20 0.34
NR4A1 P22736 1/20 0.34
NR4A2 P43354 1/20 0.34
NR4A3 Q92570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13508420 0.90 CYP1A2 (0.42) ESR1CYP2D6CYP1A2CYP3A4CYP2C9
SCHEMBL14570727 0.89 CYP1A2 (0.41) ESR1CYP2D6CYP1A2CYP3A4CYP2C9
SCHEMBL13508382 0.89 ESR1 (0.45) ESR1CYP2D6PLAUPTGS2CYP19A1
SCHEMBL13508451 0.84 PTGS1 (0.43) ESR1PLAUCYP3A4PTGS2MEN1
SCHEMBL14077314 0.83 RELA (0.36) ESR1CYP2D6PLAUCYP1A2CYP3A4
SCHEMBL13380719 0.82 ESR1 (0.44) ESR1CYP2D6PLAUPTGS2CYP19A1
SCHEMBL13508400 0.82 CYP1A2 (0.42) CYP2D6CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5877773 0.79 NR4A1 (0.48) ESR1CYP2D6CYP1A2CYP3A4CYP2C9
SCHEMBL16231505 0.79 ESR1 (0.36) ESR1CYP2D6PTGS2CYP19A1CYP11B2
SCHEMBL13511074 0.77 CYP19A1 (0.36) ESR1CYP2D6PTGS2CYP19A1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761962-B1 ORGANIC ELECTROLUMINESCENT DEVICE MERCK PATENT GMBH (DE) 2010-02-03 EP disclosed
US-20090159874-A1 Organic electroluminescent devices MERCK PATENT GMBH (DE) 2009-06-25 US disclosed
US-20090159874-A1 Organic electroluminescent devices MERCK PATENT GMBH (DE) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090159874-A1 Organic electroluminescent devices LEF1, NCS1, CRY1 ESR1 356/4885CYP2D6 1428/4885PLAU 3072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.