SCHEMBL13574288

SCHEMBL13574288

CCC(=O)c1cc(N)ccc1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
HSP90AB1 P08238 1/20 0.40
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
THRB P10828 2/20 0.38
RECQL P46063 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
PKM P14618 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 2/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
APEX1 P27695 1/20 0.38
BLM P54132 1/20 0.38
MCL1 Q07820 1/20 0.38
TNF P01375 1/20 0.38
HSPD1 P10809 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10799503 0.80 MAPT (0.55) ALOX5KMT2AMAPTMEN1THRB
SCHEMBL9041388 0.78 MAPT (0.57) ALOX5HSP90AB1KMT2AMAPTMEN1
SCHEMBL10713704 0.77 ALDH1A1 (0.60) ALOX5HSP90AB1KMT2AMAPTMEN1
SCHEMBL11989292 0.77 CASP1 (0.45) ALOX5HSP90AB1KMT2AMAPTMEN1
SCHEMBL21123646 0.76 GAA (0.57) ALOX5KMT2AMAPTMEN1KDM4E
SCHEMBL270136 0.76 GABRA1 (0.45) HSP90AB1KMT2AMAPTMEN1ALDH1A1
SCHEMBL27574494 0.75 P2RX7 (0.43) HSP90AB1KMT2AMAPTMEN1THRB
SCHEMBL27944283 0.75 HSP90AB1 (0.42) ALOX5HSP90AB1KMT2AMAPTMEN1
SCHEMBL9559750 0.74 HSP90AB1 (0.48) HSP90AB1KMT2AMAPTMEN1THRB
SCHEMBL6566640 0.73 ALDH1A1 (0.58) ALOX5MAPTKDM4EALDH1A1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155042-A1 3-SUBSTITUTED-1H-INDOLE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-12-23 WO disclosed