SCHEMBL13626507

SCHEMBL13626507

CN1CCC(N2CCN(C(=O)C3Cc4ccccc4CN3C(=O)Nc3ccc(Cl)cc3)CC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
GAA P10253 1/20 0.52
TAS1R3 Q7RTX0 2/20 0.51
TAS1R1 Q7RTX1 2/20 0.51
TAS1R2 Q8TE23 2/20 0.51
NAMPT P43490 10/20 0.49
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 1/20 0.42
PREP P48147 2/20 0.42
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CFTR P13569 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626558 0.82 MEN1 (0.53) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL76181 0.81 F10 (0.47) KCNH2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL13626559 0.80 MEN1 (0.51) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626561 0.79 MEN1 (0.47) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL4558064 0.77 TAS1R3 (0.60) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626504 0.73 NAMPT (0.51) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626549 0.73 NAMPT (0.51) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626550 0.73 NAMPT (0.51) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626560 0.73 F10 (0.52) KMT2AMEN1GAATAS1R3TAS1R1
SCHEMBL13626502 0.72 LMNA (0.58) KMT2AMEN1GAATAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed