SCHEMBL13633925

SCHEMBL13633925

COc1ccc(-c2cc(C)nn2-c2ccc(S(N)(=O)=O)cc2)cc1F

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 20/20 0.76
PTGS1 P23219 12/20 0.76
ABCB11 O95342 1/20 0.76
ALDH1A1 P00352 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL213124 0.87 PTGS2 (0.84) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL29593653 0.86 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6350722 0.86 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL24645 0.86 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL12062820 0.86 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6601340 0.85 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6344048 0.85 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6341965 0.85 PTGS2 (0.83) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL28723602 0.85 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL29355263 0.82 PTGS2 (0.73) PTGS2PTGS1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090281073-A1 HETEROAROMATIC DERIVATIVES USEFUL AS ANTICANCER AGENTS BHATTACHARYA SAMIT KUMAR 2009-11-12 US disclosed
US-20090215742-A1 AMIDE RESORCINOL COMPOUNDS PFIZER, INC. 2009-08-27 US disclosed
US-7537762-B2 Human monoclonal antibodies to activin receptor-like kinase-1 AMGEN FREMONT, INC. (US) 2009-05-26 US disclosed
US-20090111805-A1 BICYCLIC HETEROAROMATIC DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER INC. 2009-04-30 US disclosed
US-20080027011-A1 Homogeneous paste and gel formulations MERIAL LIMITED 2008-01-31 US disclosed
US-20070065444-A1 Human monoclonal antibodies to activin receptor-like kinase-1 AMGEN FREMONT INC. (US) 2007-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080027011-A1 Homogeneous paste and gel formulations EPX, CAT, PEF1 PTGS2 329/4885PTGS1 101/4885ABCB11 200/4885
US-20090111805-A1 BICYCLIC HETEROAROMATIC DERIVATIVES USEFUL AS ANTICANCER AGENTS CCNB1, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CCNY PTGS2 3711/4885PTGS1 2642/4885ABCB11 123/4885
US-20090215742-A1 AMIDE RESORCINOL COMPOUNDS HSP90AB1, HSP90AA1, HSP90AB2P PTGS2 2000/4885PTGS1 1974/4885ABCB11 29/4885
US-20070065444-A1 Human monoclonal antibodies to activin receptor-like kinase-1 SMAD3, SMAD2, ACVR1 PTGS2 4769/4885PTGS1 4487/4885ABCB11 4469/4885
US-20090281073-A1 HETEROAROMATIC DERIVATIVES USEFUL AS ANTICANCER AGENTS CCNY, TP53, CCNE1 PTGS2 3101/4885PTGS1 2342/4885ABCB11 221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.