SCHEMBL13639648

SCHEMBL13639648

N/C(=C\c1ccc(F)c(Cl)c1)c1ccc(Cl)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.43
CXCL12 P48061 1/20 0.37
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
KMT2A Q03164 3/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
MAPK1 P28482 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
CYP11B2 P19099 2/20 0.34
CASP1 P29466 2/20 0.34
CYP11B1 P15538 1/20 0.34
IDO1 P14902 1/20 0.33
DPEP1 P16444 1/20 0.33
SLC6A4 P31645 1/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12445945 0.92 NPFFR2 (0.40) TRPA1CXCL12KMT2APOLBPKM
SCHEMBL13639608 0.86 NPFFR1 (0.36) TRPA1CXCL12MAPK1CYP11B2CYP11B1
SCHEMBL12446116 0.84 GRIN1 (0.43) KMT2APOLBPKMCYP11B2MAPT
SCHEMBL12446542 0.82 MAOB (0.42) PKMMAPK1SMN1; SMN2MAOB
SCHEMBL13639614 0.80 CXCL12 (0.34) CXCL12CYP11B2CYP11B1SLC6A4MAOB
SCHEMBL13639524 0.80 DGAT1 (0.40) FLT1FLT4KDRKMT2APOLB
SCHEMBL13639667 0.79 CYP11B2 (0.36) CXCL12KMT2ACYP11B2CASP1CYP11B1
SCHEMBL2151553 0.78 POLB (0.44) TRPA1KMT2APOLBPKMMAPK1
SCHEMBL2151560 0.78 POLB (0.44) TRPA1KMT2APOLBPKMMAPK1
SCHEMBL12446099 0.73 ERN1 (0.37) CXCL12KMT2ACYP11B2CYP11B1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed