SCHEMBL13639614

SCHEMBL13639614

N/C(=C\c1cc(F)cc(Cl)c1)c1ccc(Cl)cc1F

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCL12 P48061 1/20 0.34
CYP11B2 P19099 3/20 0.33
CYP11B1 P15538 2/20 0.33
P2RX7 Q99572 2/20 0.32
SLC6A4 P31645 1/20 0.32
MAOB P27338 1/20 0.31
CYP3A4 P08684 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
TRPM5 Q9NZQ8 2/20 0.30
TRPM4 Q8TD43 1/20 0.30
P2RX1 P51575 1/20 0.30
P2RX4 Q99571 1/20 0.30
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446542 0.84 MAOB (0.42) MAOBCYP3A4NPC1RAB9A
SCHEMBL12446116 0.83 GRIN1 (0.43) CYP11B2MAOBCYP3A4NPC1RAB9A
SCHEMBL13639648 0.80 TRPA1 (0.43) CXCL12CYP11B2CYP11B1SLC6A4MAOB
SCHEMBL12445945 0.79 NPFFR2 (0.40) CXCL12CYP11B2CYP11B1SLC6A4
SCHEMBL2152623 0.78 MAPT (0.45) CYP3A4
SCHEMBL2152629 0.78 MAPT (0.45) CYP3A4
SCHEMBL13639667 0.78 CYP11B2 (0.36) CXCL12CYP11B2CYP11B1SLC6A4NPC1
SCHEMBL13639524 0.75 DGAT1 (0.40) NPC1RAB9A
SCHEMBL13639608 0.73 NPFFR1 (0.36) CXCL12CYP11B2CYP11B1CYP3A4RAB9A
SCHEMBL12446099 0.72 ERN1 (0.37) CXCL12CYP11B2CYP11B1SLC6A4RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed