SCHEMBL12445945

SCHEMBL12445945

N/C(=C\c1ccc(Cl)c(Cl)c1)c1ccc(Cl)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPFFR2 Q9Y5X5 2/20 0.40
KMT2A Q03164 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 2/20 0.38
ALDH1A1 P00352 3/20 0.37
CXCL12 P48061 1/20 0.36
TRPA1 O75762 1/20 0.36
CYP11B2 P19099 2/20 0.33
CYP11B1 P15538 1/20 0.33
CHAT P28329 1/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
SLC2A1 P11166 1/20 0.33
SLC6A4 P31645 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639648 0.92 TRPA1 (0.43) KMT2ANPSR1ALDH1A1CXCL12TRPA1
SCHEMBL13639608 0.85 NPFFR1 (0.36) NPFFR2TP53CXCL12TRPA1CYP11B2
SCHEMBL12446116 0.83 GRIN1 (0.43) KMT2AALDH1A1CYP11B2CHATPOLB
SCHEMBL12446542 0.81 MAOB (0.42) PKMMAPK1SMN1; SMN2
SCHEMBL13639614 0.79 CXCL12 (0.34) CXCL12CYP11B2CYP11B1SLC6A4
SCHEMBL30006425 0.78 ALDH1A1 (0.42) KMT2ANPSR1ALDH1A1POLBPKM
SCHEMBL2151442 0.78 ALDH1A1 (0.42) KMT2ANPSR1ALDH1A1POLBPKM
SCHEMBL13639524 0.78 DGAT1 (0.40) KMT2ANPSR1ALDH1A1POLBPKM
SCHEMBL2151454 0.78 ALDH1A1 (0.42) KMT2ANPSR1ALDH1A1POLBPKM
SCHEMBL13639667 0.78 CYP11B2 (0.36) KMT2ANPSR1ALDH1A1CXCL12CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed
WO-2011098398-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-18 WO disclosed