SCHEMBL13639608

SCHEMBL13639608

N/C(=C\c1ccc(C(F)(F)F)c(Cl)c1)c1ccc(Cl)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPFFR1 Q9GZQ6 2/20 0.36
NPFFR2 Q9Y5X5 2/20 0.36
SCN9A Q15858 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
CXCL12 P48061 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TRPA1 O75762 1/20 0.33
CYP3A4 P08684 3/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP3A5 P20815 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KIF11 P52732 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639648 0.86 TRPA1 (0.43) CYP11B1CYP11B2CXCL12MAPTSMN1; SMN2
SCHEMBL12445945 0.85 NPFFR2 (0.40) NPFFR2CYP11B1CYP11B2CXCL12TP53
SCHEMBL2152020 0.81 ALDH1A1 (0.38) CYP11B1CYP11B2MAPTSMN1; SMN2CYP3A4
SCHEMBL2152012 0.81 ALDH1A1 (0.38) CYP11B1CYP11B2MAPTSMN1; SMN2CYP3A4
SCHEMBL12446116 0.77 GRIN1 (0.43) CYP11B2MAPTRAB9ASMN1; SMN2CYP3A4
SCHEMBL12446542 0.75 MAOB (0.42) RAB9ASMN1; SMN2CYP3A4MAPK1TDP1
SCHEMBL13639614 0.73 CXCL12 (0.34) CYP11B1CYP11B2CXCL12RAB9ACYP3A4
SCHEMBL13639524 0.73 DGAT1 (0.40) MAPTRAB9ASMN1; SMN2KDM4EGRIK1
SCHEMBL13639667 0.72 CYP11B2 (0.36) CYP11B1CYP11B2CXCL12MAPTRAB9A
SCHEMBL29403188 0.69 TSHR (0.62) TP53RAB9ACYP3A4TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed