SCHEMBL13639667

SCHEMBL13639667

N/C(=C\c1cc(Cl)ccc1F)c1ccc(Cl)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.36
CYP11B1 P15538 2/20 0.36
SLC6A4 P31645 1/20 0.35
ERN1 O75460 1/20 0.34
CXCL12 P48061 1/20 0.34
GRIN2D O15399 2/20 0.33
GRIN3B O60391 2/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2A Q12879 2/20 0.33
GRIN2B Q13224 2/20 0.33
GRIN2C Q14957 2/20 0.33
GRIN3A Q8TCU5 2/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
DGAT1 O75907 1/20 0.33
KDM4E B2RXH2 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639623 0.84 KDM4E (0.52) CYP11B2CYP11B1SLC6A4ERN1CXCL12
SCHEMBL12446099 0.83 ERN1 (0.37) CYP11B2CYP11B1SLC6A4ERN1CXCL12
SCHEMBL13639590 0.79 CYP11B2 (0.32) CYP11B2CYP11B1SLC6A4ERN1
SCHEMBL13639648 0.79 TRPA1 (0.43) CYP11B2CYP11B1SLC6A4CXCL12MAPT
SCHEMBL12446116 0.79 GRIN1 (0.43) CYP11B2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12445945 0.78 NPFFR2 (0.40) CYP11B2CYP11B1SLC6A4CXCL12MAPT
SCHEMBL13639614 0.78 CXCL12 (0.34) CYP11B2CYP11B1SLC6A4CXCL12NPC1
SCHEMBL12446542 0.76 MAOB (0.42) GRIN2BSMN1; SMN2NPC1RAB9ANFE2L2
SCHEMBL2151880 0.76 CYP1A2 (0.44) CYP11B2CYP11B1MAPTNPSR1KDM4E
SCHEMBL2151888 0.76 CYP1A2 (0.44) CYP11B2CYP11B1MAPTNPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed