SCHEMBL1365293

SCHEMBL1365293

CC(C)(C)OC(=O)N1CCCCC(N)C1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.55
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
EPHX1 P07099 1/20 0.49
PREP P48147 2/20 0.47
USP2 O75604 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RECQL P46063 1/20 0.42
NR1H2 P55055 1/20 0.42
PDE4B Q07343 1/20 0.42
BACE1 P56817 2/20 0.42
CTSD P07339 1/20 0.42
KDM4E B2RXH2 1/20 0.42
THRB P10828 1/20 0.42
ABL1 P00519 1/20 0.41
RIN1 Q13671 1/20 0.41
USP30 Q70CQ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1563471 1.00 HPGD (0.55) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL16041868 1.00 HPGD (0.55) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL31045792 0.98 HPGD (0.57) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL18391127 0.98 HPGD (0.57) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL21890138 0.98 HPGD (0.57) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL376485 0.95 MAPT (0.55) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL181567 0.95 MAPT (0.55) HPGDMAPTMEN1ALDH1A1KMT2A
SCHEMBL181566 0.95 MAPT (0.55) HPGDMAPTMEN1ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL641221 0.94 MAPT (0.53) HPGDMAPTMEN1ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL9104390 0.94 MAPT (0.53) HPGDMAPTMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 226 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116042560-A Mutant of recombinant aminotransferase and application thereof 清华大学 2023-05-02 CN claimed
US-12570672-B2 Macrocyclic compounds and methods of use AMGEN INC. 2026-03-10 US disclosed
US-20250320228-A1 PYRIDO[3,2-D]PYRIMIDINES AS HPK1 INHIBITORS MERCK PATENT GMBH (DE) 2025-10-16 US disclosed
US-20250304599-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2025-10-02 US disclosed
EP-4598921-A1 MACROCYCLIC KRAS INHIBITORS AND METHODS OF USE Amgen Inc. (US) 2025-08-13 EP disclosed
US-20250236631-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2025-07-24 US disclosed
US-20250115619-A1 BRIDGED TRICYCLIC CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2025-04-10 US disclosed
US-20250099442-A1 COMPOUNDS FOR USE IN TREATING NEUROLOGICAL DISORDERS PROTHENA BIOSCIENCES INC 2025-03-27 US disclosed
CN-119546604-A Pyrido [3,2-D ] pyrimidines as HPK1 inhibitors 默克专利有限公司 2025-02-28 CN disclosed
EP-4507789-A1 PYRIDO[3,2-D]PYRIMIDINES AS HPK1 INHIBITORS Merck Patent GmbH (DE) 2025-02-19 EP disclosed
EP-2046793-A2 FUSED PYRIMIDO COMPOUNDS AstraZeneca AB (SE) 2009-04-15 EP disclosed
US-20090054396-A1 SUBSTITUTED THIOPHENES AND USES THEREOF ASTRAZENECA AB (SE) 2009-02-26 US disclosed
EP-1660474-B1 SUBSTITUTED THIOPHENES AND USES THEREOF ASTRAZENECA AB (SE) 2008-10-29 EP disclosed
US-7423061-B2 Substitute thiophenes and uses thereof ASTRAZENECA AB (SE) 2008-09-09 US disclosed
WO-2008003958-A2 FUSED PYRIMIDO COMPOUNDS ASTRAZENECA AB (SE) 2008-01-10 WO disclosed
US-20080009482-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2008-01-10 US disclosed
US-20070010556-A1 Thiophene derivatives as chk 1 inhibitors ASTRAZENECA AB (SE) 2007-01-11 US disclosed
US-20060281666-A1 Substitute thiophenes and uses therof ASTRAZENECA AB (SE) 2006-12-14 US disclosed
US-20050182040-A1 Benzamide derivatives DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2005-08-18 US disclosed
EP-1500643-A1 BENZAMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2005-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250115619-A1 BRIDGED TRICYCLIC CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE ZYX, CCNY, NCAPD3 HPGD 550/4885MAPT 1576/4885MEN1 3930/4885
US-20250320228-A1 PYRIDO[3,2-D]PYRIMIDINES AS HPK1 INHIBITORS PDXK, PPIP5K2, IP6K1 HPGD 162/4885MAPT 3349/4885MEN1 2014/4885
US-20250236631-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE KRAS, NRAS, HRAS HPGD 1367/4885MAPT 4614/4885MEN1 166/4885
US-20070010556-A1 Thiophene derivatives as chk 1 inhibitors CHEK1, CHKA, CHEK2 HPGD 3165/4885MAPT 3514/4885MEN1 3068/4885
US-12570672-B2 Macrocyclic compounds and methods of use KRAS, NRAS, BRAF HPGD 2567/4885MAPT 3706/4885MEN1 34/4885
US-20250304599-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE KRAS, NRAS, HRAS HPGD 1367/4885MAPT 4614/4885MEN1 166/4885
US-20250099442-A1 COMPOUNDS FOR USE IN TREATING NEUROLOGICAL DISORDERS DYRK2, DYRK1A, DYRK1B HPGD 2718/4885MAPT 36/4885MEN1 3098/4885
US-20080009482-A1 NOVEL COMPOUNDS CYP11B2, CYP11B1, CYP46A1 HPGD 307/4885MAPT 2200/4885MEN1 1408/4885
US-20090054396-A1 SUBSTITUTED THIOPHENES AND USES THEREOF TPMT, ABCG2, TYMP HPGD 808/4885MAPT 2490/4885MEN1 1076/4885
US-20060281666-A1 Substitute thiophenes and uses therof TYMP, TPMT, MGMT HPGD 1838/4885MAPT 1633/4885MEN1 1011/4885
US-20050182040-A1 Benzamide derivatives ROCK1, ROCK2, NHERF1 HPGD 339/4885MAPT 4237/4885MEN1 1993/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.