SCHEMBL13680491

SCHEMBL13680491

Cc1csc(-c2ccc(C(=O)O)nc2)n1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
HPGDS O60760 2/20 0.50
CYP2E1 P05181 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2A6 P11509 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2B6 P20813 1/20 0.49
P4HA1 P13674 1/20 0.42
MIF P14174 1/20 0.42
P4HTM Q9NXG6 1/20 0.42
ECE1 P42892 2/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
TGFBR1 P36897 2/20 0.41
KDM4E B2RXH2 1/20 0.41
AOC3 Q16853 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680540 0.84 DYRK1A (0.52) ALDH1A1HPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL6840352 0.79 CYP3A4 (0.64) ALDH1A1HPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL13680478 0.78 KDM4E (0.62) ALDH1A1NPC1POLBRAB9AKDM4E
SCHEMBL13680530 0.74 CYP2A6 (0.54) ALDH1A1CYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL13680949 0.74 HPGDS (0.43) ALDH1A1HPGDSKDM4E
SCHEMBL13731115 0.74 P4HTM (0.64) ALDH1A1CYP3A4P4HA1MIFP4HTM
SCHEMBL8198560 0.74 CYP3A4 (0.60) ALDH1A1CYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL2079765 0.74 HPGDS (0.62) ALDH1A1HPGDSKDM4E
SCHEMBL31340947 0.73 HPGDS (0.47) ALDH1A1HPGDSECE1KDM4E
SCHEMBL13680742 0.73 CYP2E1 (0.45) ALDH1A1HPGDSCYP2E1CYP3A4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed