SCHEMBL13680658

SCHEMBL13680658

Cc1cccc(-c2cnc(N(C)C)cn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.47
ACHE P22303 1/20 0.47
IDO1 P14902 1/20 0.46
METAP2 P50579 1/20 0.46
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
KDM1A O60341 1/20 0.44
KMO O15229 2/20 0.41
GRIN2B Q13224 1/20 0.41
ATR Q13535 1/20 0.40
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
EGFR P00533 1/20 0.40
NISCH Q9Y2I1 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3422110 0.86 IDO1 (0.58) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL23601607 0.79 KDM1A (0.53) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL8265012 0.78 APP (0.50) HSD17B1HSD17B2GRIN2BEGFRNPC1
SCHEMBL16826157 0.76 KDM1A (0.50) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL13680659 0.75 RAB9A (0.66) IDO1METAP2KDM1AKMONISCH
SCHEMBL23601695 0.73 BCHE (0.47) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL23601693 0.73 KDR (0.48) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL24636033 0.73 BCHE (0.47) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL12973163 0.73 HSD17B1 (0.59) BCHEACHEIDO1METAP2HSD17B1
SCHEMBL12797772 0.73 CYP3A4 (0.59) BCHEACHEIDO1METAP2HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed