SCHEMBL13680701

SCHEMBL13680701

Cc1ccc(-c2ccc(C(N)=S)cc2)o1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.53
TOP2B Q02880 3/20 0.53
NQO2 P16083 8/20 0.48
ALDH1A1 P00352 1/20 0.48
TOP1 P11387 1/20 0.48
HPGD P15428 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PRMT1 Q99873 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
GSK3B P49841 3/20 0.45
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680696 0.83 GSK3B (0.43) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL13680503 0.81 GSK3B (0.62) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL13681315 0.81 TOP2A (0.44) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL23197679 0.79 TDP1 (0.56) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL13680703 0.79 ALDH1A1 (0.46) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL13680707 0.79 MAPT (0.40) TOP2ATOP2BNQO2ALDH1A1TOP1
SCHEMBL13680705 0.77 ALDH1A1 (0.48) ALDH1A1HPGDHSD17B10TDP1SMN1; SMN2
SCHEMBL13680452 0.76 GSK3B (0.61) NQO2ALDH1A1HPGDGSK3BSMN1; SMN2
SCHEMBL13680465 0.76 GSK3B (0.61) NQO2ALDH1A1HPGDTDP1GSK3B
SCHEMBL14046637 0.75 NQO2 (0.44) TOP2ATOP2BNQO2ALDH1A1TOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed