SCHEMBL13680703

SCHEMBL13680703

Cc1ccc(-c2ccc(C(=S)N(C)C)cc2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MAPT P10636 3/20 0.46
GSK3B P49841 5/20 0.38
HPGD P15428 5/20 0.38
HSD17B10 Q99714 4/20 0.38
TOP2A P11388 3/20 0.38
TOP2B Q02880 3/20 0.38
NQO2 P16083 3/20 0.38
PRMT1 Q99873 2/20 0.38
TOP1 P11387 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
BACE1 P56817 1/20 0.38
GAA P10253 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680696 0.80 GSK3B (0.43) ALDH1A1MAPTGSK3BHPGDHSD17B10
SCHEMBL13680494 0.79 ALDH1A1 (0.46) ALDH1A1MAPTGSK3BHPGDNQO2
SCHEMBL13680701 0.79 TOP2A (0.53) ALDH1A1MAPTGSK3BHPGDHSD17B10
SCHEMBL23197679 0.77 TDP1 (0.56) ALDH1A1MAPTGSK3BHPGDHSD17B10
SCHEMBL13680707 0.76 MAPT (0.40) ALDH1A1MAPTGSK3BHPGDHSD17B10
SCHEMBL13681315 0.75 TOP2A (0.44) ALDH1A1MAPTGSK3BHPGDHSD17B10
SCHEMBL13680452 0.73 GSK3B (0.61) ALDH1A1MAPTGSK3BHPGDNQO2
SCHEMBL13680465 0.73 GSK3B (0.61) ALDH1A1MAPTGSK3BHPGDNQO2
SCHEMBL13680998 0.72 ALDH1A1 (0.41) ALDH1A1MAPTHPGDHSD17B10PRMT1
SCHEMBL13680503 0.71 GSK3B (0.62) ALDH1A1GSK3BHPGDHSD17B10TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed