SCHEMBL13680760

SCHEMBL13680760

CNc1ncc(-c2nc(C)cs2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2E1 P05181 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2B6 P20813 1/20 0.38
KDR P35968 1/20 0.36
LMNA P02545 1/20 0.35
LIMK1 P53667 1/20 0.35
SPHK2 Q9NRA0 1/20 0.35
SPHK1 Q9NYA1 1/20 0.35
RAB9A P51151 5/20 0.34
NPC1 O15118 4/20 0.34
FDPS P14324 1/20 0.34
CDK2 P24941 2/20 0.34
SRC P12931 1/20 0.34
ZAP70 P43403 1/20 0.34
SYK P43405 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK1 P06493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680759 0.76 BACE1 (0.49) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL13680737 0.73 ADORA2A (0.39) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL13680758 0.73 DYRK1A (0.43) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL13681065 0.73 ALDH1A1 (0.33) LMNALIMK1RAB9ACDK2CCNT1
SCHEMBL13681281 0.72 LOXL2 (0.41) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL259247 0.69
SCHEMBL13680746 0.69 CYP3A4 (0.47) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL22631683 0.69 PDE10A (0.36) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6
SCHEMBL13680697 0.69 KDR (0.51) CYP3A4CYP2C9CYP2A6KDRLMNA
SCHEMBL18157874 0.69 SMN1; SMN2 (0.55) PDE10ACYP3A4CYP2C9CYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed